SCHEMBL1386352

SCHEMBL1386352

CC(=O)N1CCN(C(C)NC(=O)c2cccc(-c3cnc(N)c(OCc4cccc(F)c4C(F)(F)F)n3)c2)CC1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ATR Q13535 11/20 0.36
PIK3CA P42336 2/20 0.36
PIK3CD O00329 1/20 0.36
PIK3CG P48736 1/20 0.36
LDHB P07195 3/20 0.35
LDHA P00338 2/20 0.35
MAPK1 P28482 2/20 0.35
CSF1R P07333 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL488293 0.86 ATR (0.48) ATRCSF1R
SCHEMBL30454557 0.81 ATR (0.51) ATRPIK3CAPIK3CDPIK3CGCSF1R
SCHEMBL488175 0.81 ATR (0.51) ATRPIK3CAPIK3CDPIK3CGCSF1R
SCHEMBL488637 0.79 LDHA (0.46) ATRPIK3CAPIK3CDPIK3CGLDHB
SCHEMBL30453342 0.79 LDHA (0.46) ATRPIK3CAPIK3CDPIK3CGLDHB
SCHEMBL488441 0.78 ATR (0.51) ATR
SCHEMBL30454216 0.78 ATR (0.51) ATR
SCHEMBL10216349 0.77 MAP4K4 (0.52) ATRPIK3CDPIK3CG
SCHEMBL488626 0.76 KCNH2 (0.56) ATR
SCHEMBL30454874 0.76 KCNH2 (0.56) ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4695588-B2 2011-06-08 JP claimed
JP-2006519232-A 2006-08-24 JP claimed
EP-1603570-A2 AMINOHETEROARYL COMPOUNDS AS PROTEIN KINASE INHIBITORS Sugen, Inc. (US) 2005-12-14 EP claimed
WO-2004076412-A2 AMINOHETEROARYL COMPOUNDS AS PROTEIN KINASE INHIBITORS SUGEN, INC. (US) 2004-09-10 WO claimed