SCHEMBL30454557

SCHEMBL30454557

CN1CCN(C(=O)c2cccc(-c3cnc(N)c(OCc4cccc(F)c4C(F)(F)F)n3)c2)CC1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ATR Q13535 5/20 0.51
KCNH2 Q12809 5/20 0.47
FYN P06241 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
ERN1 O75460 1/20 0.43
KDM4E B2RXH2 1/20 0.42
PIK3CD O00329 1/20 0.42
PIK3CA P42336 1/20 0.42
PIK3CB P42338 1/20 0.42
PIK3CG P48736 1/20 0.42
ADORA2A P29274 1/20 0.42
AURKA O14965 1/20 0.41
AURKB Q96GD4 1/20 0.41
NTRK1 P04629 1/20 0.41
ABL1 P00519 1/20 0.41
BCR P11274 1/20 0.41
CSF1R P07333 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL488175 1.00 ATR (0.51) ATRKCNH2FYNL3MBTL1ERN1
SCHEMBL30454874 0.93 KCNH2 (0.56) ATRKCNH2AURKAAURKBABL1
SCHEMBL488626 0.93 KCNH2 (0.56) ATRKCNH2AURKAAURKBABL1
SCHEMBL30454051 0.87 ATR (0.54) ATRL3MBTL1CSF1R
SCHEMBL488768 0.87 ATR (0.54) ATRL3MBTL1CSF1R
SCHEMBL488637 0.84 LDHA (0.46) ATRPIK3CDPIK3CAPIK3CGCSF1R
SCHEMBL30453342 0.84 LDHA (0.46) ATRPIK3CDPIK3CAPIK3CGCSF1R
SCHEMBL488293 0.83 ATR (0.48) ATRABL1BCRCSF1R
SCHEMBL488822 0.82 ATR (0.53) ATRKCNH2FYNERN1ADORA2A
SCHEMBL30452937 0.82 ATR (0.53) ATRKCNH2FYNERN1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113181362-B Medicament for preventing and/or treating amyotrophic lateral sclerosis 国立大学法人京都大学 2023-06-13 CN disclosed