SCHEMBL13867671

SCHEMBL13867671

CN[C@@H]1CCCC[C@H]1CN1CC(=O)N[C@@H](Cc2ccc(F)cc2)C1=O

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
OPRK1 P41145 2/20 0.38
CCR3 P51677 14/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13867668 0.84 HDAC6 (0.41) HDAC6HDAC1HDAC8OPRK1
SCHEMBL3878037 0.84 HDAC6 (0.41) HDAC6HDAC1HDAC8OPRK1
SCHEMBL3878033 0.84 HDAC6 (0.41) HDAC6HDAC1HDAC8OPRK1
SCHEMBL7112217 0.80 HDAC6 (0.46) HDAC6HDAC1HDAC8OPRK1CCR3
SCHEMBL3878046 0.80 HDAC6 (0.46) HDAC6HDAC1HDAC8OPRK1CCR3
SCHEMBL3885462 0.80 CCR3 (0.63) CCR3
SCHEMBL13867601 0.79 CCR3 (0.43) CCR3
SCHEMBL3891784 0.79 CCR3 (0.66) CCR3
SCHEMBL3888971 0.77 CCR3 (0.66) CCR3
SCHEMBL3889303 0.77 CCR3 (0.66) CCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7514430-B2 Piperizinones as modulators of chemokine receptor activity BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2009-04-07 US disclosed