SCHEMBL13868385

SCHEMBL13868385

CC(=O)N1C=CN(Cc2ccccc2)C(=O)C1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.47
DRD4 P21917 1/20 0.47
DRD3 P35462 1/20 0.47
BRD4 O60885 5/20 0.45
BRS3 P32247 1/20 0.44
ALDH1A1 P00352 2/20 0.41
CYP2D6 P10635 2/20 0.41
POLB P06746 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
ACE P12821 1/20 0.40
TSHR P16473 2/20 0.40
LMNA P02545 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HPGD P15428 1/20 0.40
NPC1 O15118 1/20 0.40
GLA P06280 1/20 0.40
MAPT P10636 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3904629 0.85 HTT (0.47) DRD2DRD4DRD3ALDH1A1POLB
SCHEMBL14547790 0.80 CACNA1G (0.45) DRD2DRD4DRD3ALDH1A1CYP2C19
SCHEMBL2895538 0.74 HTT (0.43) DRD2DRD4DRD3ALDH1A1LMNA
SCHEMBL3908131 0.70 BRD4 (0.55) BRD4ALDH1A1CYP2D6POLBCYP2C9
SCHEMBL27477427 0.70 HPGD (0.49) ALDH1A1CYP2D6POLBCYP2C9CYP2C19
SCHEMBL29157597 0.69 HPGD (0.45) ALDH1A1CYP2D6POLBCYP2C9CYP2C19
SCHEMBL13868376 0.69 BRS3 (0.52) BRD4BRS3ALDH1A1ACETSHR
SCHEMBL5807696 0.69 CACNA1G (0.45) DRD2DRD4DRD3BRD4BRS3
Acetic Acid SCHEMBL28332665 0.68 CYP2D6 (0.49) BRD4ALDH1A1CYP2D6POLBCYP2C9
SCHEMBL13868378 0.68 BRD4 (0.60) BRD4BRS3ALDH1A1TSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7517532-B2 Dihydroxypyridopyrazine-1,6-dione compounds useful as HIV integrase inhibitors MERCK & CO., INC. (US) 2009-04-14 US disclosed