SCHEMBL13874367

SCHEMBL13874367

CC(C)Oc1nnc(-c2cnc3ccc(C4=CN=C4c4ccc(F)cc4F)cn23)o1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 7/20 0.42
PIK3R1 P27986 6/20 0.42
MAPK14 Q16539 9/20 0.38
TGFBR1 P36897 4/20 0.37
MTOR P42345 2/20 0.37
PIK3CD O00329 1/20 0.37
PIK3CB P42338 1/20 0.37
PIK3CG P48736 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13874593 0.87 PIK3CA (0.46) PIK3CAPIK3R1MAPK14TGFBR1MTOR
SCHEMBL13874185 0.82 MAPK14 (0.42) PIK3CAPIK3R1MAPK14TGFBR1MTOR
SCHEMBL13874536 0.78 NOTUM (0.40) PIK3CAPIK3R1MAPK14TGFBR1MTOR
SCHEMBL3846792 0.78 TGFBR1 (0.38) PIK3CAPIK3R1MAPK14TGFBR1MTOR
SCHEMBL13874443 0.76 PIK3CA (0.39) PIK3CAPIK3R1MAPK14TGFBR1MTOR
SCHEMBL3847272 0.73 PIK3CA (0.46) PIK3CAPIK3R1MAPK14TGFBR1MTOR
SCHEMBL13874626 0.72 MAPK14 (0.34) PIK3CAPIK3R1MAPK14TGFBR1MTOR
SCHEMBL3848709 0.71 PIK3CA (0.44) PIK3CAPIK3R1MTOR
SCHEMBL3847818 0.70 PIK3CA (0.45) PIK3CAPIK3R1MAPK14TGFBR1MTOR
SCHEMBL3847367 0.69 PIK3CA (0.42) PIK3CAPIK3R1MAPK14TGFBR1MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed