SCHEMBL13874451

SCHEMBL13874451

CSc1ccc(C(=O)C2CCNCC2)s1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.51
LIG1 P18858 1/20 0.51
MEN1 O00255 1/20 0.45
CYP2D6 P10635 1/20 0.45
KMT2A Q03164 1/20 0.45
PLAU P00749 1/20 0.44
KHK P50053 2/20 0.38
HRH3 Q9Y5N1 1/20 0.38
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
HTR3A P46098 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
TSHR P16473 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3847567 0.98 PKM (0.50) PKMLIG1MEN1CYP2D6KMT2A
Hydrochloric Acid SCHEMBL224845 0.75 MEN1 (0.47) MEN1CYP2D6KMT2AHRH3HTR3E
Hydrochloric Acid SCHEMBL229437 0.75 MEN1 (0.47) MEN1CYP2D6KMT2AHRH3HTR3E
SCHEMBL6206003 0.71 MEN1 (0.41) MEN1CYP2D6KMT2ATSHRALDH1A1
Hydrochloric Acid SCHEMBL6207103 0.71 MEN1 (0.43) MEN1CYP2D6KMT2ATSHRSLC6A2
SCHEMBL13874024 0.70 MEN1 (0.66) MEN1CYP2D6KMT2AKHKALDH1A1
SCHEMBL13874464 0.70 SLC6A2 (0.35) PKMLIG1PLAUSLC6A2SLC6A4
SCHEMBL9373389 0.69 PKM (0.70) PKMLIG1PLAUTSHRNR1D1
SCHEMBL2723219 0.69 PKM (1.00) PKMLIG1MEN1KMT2APLAU
Tert-Butyl Formate SCHEMBL28779357 0.69 MEN1 (0.39) MEN1CYP2D6KMT2AHRH3HTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP disclosed