SCHEMBL1388331

SCHEMBL1388331

Nc1ncc(-c2cccc(F)c2)c(N)n1

nearest known ligand 0.67

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DHFR P00374 6/20 0.67
ADORA1 P30542 5/20 0.49
ADORA2A P29274 2/20 0.47
MAP4K4 O95819 2/20 0.46
CCNT1 O60563 1/20 0.45
CCNA2 P20248 1/20 0.45
CDK2 P24941 1/20 0.45
CDK9 P50750 1/20 0.45
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
MAPT P10636 1/20 0.45
KMT2A Q03164 1/20 0.45
CHEK2 O96017 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27974551 0.85 DHFR (0.49) DHFRADORA1ADORA2AMAP4K4KDM4E
SCHEMBL30401146 0.83 DHFR (0.71) DHFRADORA1ADORA2AMAP4K4
SCHEMBL1388358 0.83 DHFR (0.71) DHFRADORA1ADORA2AMAP4K4
SCHEMBL4613214 0.82 DHFR (0.53) DHFRADORA1
SCHEMBL27631899 0.81 DHFR (0.69) DHFRADORA1ADORA2A
SCHEMBL20150236 0.80 ADORA1 (0.51) DHFRADORA1ADORA2AMAPT
SCHEMBL1388335 0.80 DHFR (0.67) DHFRADORA1ADORA2AKDM4EMEN1
SCHEMBL1388276 0.80 ADORA1 (0.70) DHFRADORA1ADORA2AMAP4K4CDK9
SCHEMBL29913330 0.80 DHFR (1.00) DHFRADORA1ADORA2AMAP4K4
SCHEMBL1116404 0.80 ADORA1 (0.70) DHFRADORA1ADORA2AMAP4K4CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-H08504798-A 1996-05-21 JP claimed
WO-1994014780-A1 PYRIMIDINE, PYRIDINE, PTERIDINONE AND INDAZOLE DERIVATIVES AS ENZYME INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1994-07-07 WO claimed
WO-1994014780-A1 PYRIMIDINE, PYRIDINE, PTERIDINONE AND INDAZOLE DERIVATIVES AS ENZYME INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1994-07-07 WO disclosed