SCHEMBL29913330

SCHEMBL29913330

Nc1ncc(-c2cccc(Cl)c2)c(N)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DHFR P00374 7/20 1.00
ADORA1 P30542 2/20 0.70
ADORA2A P29274 1/20 0.70
PTPN11 Q06124 1/20 0.54
TDO2 P48775 1/20 0.51
MAP4K4 O95819 2/20 0.51
FGFR1 P11362 1/20 0.50
SRC P12931 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1388562 1.00 DHFR (1.00) DHFRADORA1ADORA2APTPN11TDO2
SCHEMBL30401146 0.83 DHFR (0.71) DHFRADORA1ADORA2AMAP4K4FGFR1
SCHEMBL1388358 0.83 DHFR (0.71) DHFRADORA1ADORA2AMAP4K4FGFR1
SCHEMBL1388590 0.82 DHFR (0.70) DHFRADORA1ADORA2AMAP4K4FGFR1
SCHEMBL27631899 0.81 DHFR (0.69) DHFRADORA1ADORA2A
SCHEMBL30488016 0.80 ADORA1 (0.70) DHFRADORA1ADORA2AMAP4K4FGFR1
SCHEMBL1388335 0.80 DHFR (0.67) DHFRADORA1ADORA2AFGFR1
SCHEMBL1388331 0.80 DHFR (0.67) DHFRADORA1ADORA2AMAP4K4
SCHEMBL1388276 0.80 ADORA1 (0.70) DHFRADORA1ADORA2AMAP4K4FGFR1
SCHEMBL1116404 0.80 ADORA1 (0.70) DHFRADORA1ADORA2AMAP4K4FGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220289686-A1 COMPOSITIONS OF NRF2 INHIBITING AGENTS AND METHODS OF USE THEREOF WASHINGTON UNIVERSITY 2022-09-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220289686-A1 COMPOSITIONS OF NRF2 INHIBITING AGENTS AND METHODS OF USE THEREOF KEAP1, GSTK1, NFE2L2 DHFR 1701/4885ADORA1 3948/4885ADORA2A 2453/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.