SCHEMBL13891719

SCHEMBL13891719

Cc1ccccc1-c1nc(N2CCCN(C)CC2)nc2c1C(=O)N(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)CCCO2

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 17/20 0.48
CASP1 P29466 1/20 0.37
CASP5 P51878 1/20 0.37
BRAF P15056 1/20 0.34
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13891620 0.90 TACR1 (0.43) TACR1CASP1CASP5
SCHEMBL6508415 0.89 TACR1 (0.44) TACR1
SCHEMBL29373661 0.89 TACR1 (0.44) TACR1
SCHEMBL13891688 0.87 TACR1 (0.41) TACR1CASP1CASP5
SCHEMBL15680049 0.85 TACR1 (0.41) TACR1
SCHEMBL13891718 0.85 TACR1 (0.40) TACR1BRAFROCK2ROCK1
SCHEMBL13891760 0.83 TACR1 (0.41) TACR1ROCK2ROCK1
SCHEMBL13891689 0.83 TACR1 (0.35) TACR1ROCK2ROCK1
SCHEMBL13891717 0.82 ADRB2 (0.43) TACR1CASP1CASP5ROCK2ROCK1
SCHEMBL13891621 0.82 TACR1 (0.38) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1473295-B1 FUSED BICYCLIC PYRIMIDINE DERIVATIVES KYORIN SEIYAKU KK (JP) 2009-04-01 EP disclosed