SCHEMBL13891767

SCHEMBL13891767

CC(=O)N1CCN(c2nc3c(c(-c4ccccc4C)n2)C(=O)N(Cc2ccccc2)CCCO3)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 4/20 0.40
SMO Q99835 2/20 0.39
ACHE P22303 2/20 0.38
PIK3R1 P27986 1/20 0.38
MTOR P42345 1/20 0.38
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
NCF1 P14598 1/20 0.37
HTT P42858 2/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
GBA1 P04062 2/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13891721 0.94 HTT (0.37) P2RX3SMOPIK3R1MTORHTT
SCHEMBL6508415 0.90 TACR1 (0.44) P2RX3PIK3R1MTOR
SCHEMBL29373661 0.90 TACR1 (0.44) P2RX3PIK3R1MTOR
SCHEMBL13891620 0.88 TACR1 (0.43) P2RX3
SCHEMBL15680049 0.87 TACR1 (0.41) P2RX3PIK3R1MTOR
SCHEMBL13891686 0.81 MAPT (0.35) PDE4APDE4BPDE4CPDE4DMEN1
SCHEMBL13891740 0.79 TLR7 (0.36) MEN1KMT2AL3MBTL1CYP2C9
SCHEMBL13891719 0.78 TACR1 (0.48)
SCHEMBL5527526 0.76 TACR1 (0.43)
SCHEMBL5230814 0.76 TACR1 (0.44) P2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1473295-B1 FUSED BICYCLIC PYRIMIDINE DERIVATIVES KYORIN SEIYAKU KK (JP) 2009-04-01 EP disclosed