SCHEMBL13891740

SCHEMBL13891740

Cc1ccccc1-c1nc(S(C)(=O)=O)nc2c1C(=O)N(Cc1ccccc1)CCCO2

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 1/20 0.36
SDHB P21912 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
KCNH2 Q12809 1/20 0.34
GRM2 Q14416 1/20 0.34
MAPK14 Q16539 1/20 0.33
DGAT1 O75907 1/20 0.33
CLPP Q16740 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
BACE1 P56817 1/20 0.32
P2RX7 Q99572 1/20 0.32
DHPS P49366 1/20 0.32
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
TSHR P16473 1/20 0.31
CYP2C19 P33261 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13891686 0.85 MAPT (0.35) MEN1KMT2AKCNH2GRM2MAPK14
SCHEMBL13891616 0.83 SDHB (0.40) SDHB
SCHEMBL13891767 0.79 P2RX3 (0.40) MEN1KMT2AL3MBTL1CYP2C9
SCHEMBL13891759 0.79 TACR1 (0.37) P2RX7
SCHEMBL13891702 0.78 KDM4E (0.41) SDHBMEN1KMT2AL3MBTL1TSHR
SCHEMBL13891760 0.74 TACR1 (0.41)
SCHEMBL5232743 0.73 TACR1 (0.40) SDHBL3MBTL1CYP3A4CYP2D6
SCHEMBL13891721 0.73 HTT (0.37) MEN1KMT2AL3MBTL1CYP2C9
SCHEMBL13891738 0.73 TACR1 (0.41) MEN1KMT2ACYP3A4CYP2D6CYP2C9
SCHEMBL5225462 0.73 SDHB (0.40) SDHB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1473295-B1 FUSED BICYCLIC PYRIMIDINE DERIVATIVES KYORIN SEIYAKU KK (JP) 2009-04-01 EP disclosed