SCHEMBL13894111

SCHEMBL13894111

CN(C)c1ccc(C(=O)Nc2cccc(-c3c[nH]c(=O)c(Nc4ccc(C(=O)N5CCC(N(C)C)CC5)cn4)c3)c2CO)cc1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BTK Q06187 15/20 0.53
CLK2 P49760 1/20 0.53
ITK Q08881 3/20 0.42
KIT P10721 2/20 0.42
SRC P12931 2/20 0.42
FLT3 P36888 2/20 0.42
CDK4 P11802 1/20 0.38
CDK6 Q00534 1/20 0.38
CCNA2 P20248 1/20 0.37
CDK2 P24941 1/20 0.37
TTK P33981 1/20 0.37
AURKB Q96GD4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12602943 0.88 BTK (0.69) BTKCLK2
SCHEMBL13894038 0.83 ITK (0.47) BTKCLK2ITKKITSRC
SCHEMBL13894051 0.83 BTK (0.67) BTKCLK2SRC
SCHEMBL13894115 0.82 BTK (0.63) BTKCLK2ITKSRC
SCHEMBL13894012 0.82 BTK (0.78) BTKCLK2ITKSRCFLT3
SCHEMBL13894023 0.82 BTK (0.67) BTKCLK2
SCHEMBL13894124 0.81 BTK (0.65) BTKCLK2SRC
SCHEMBL13894117 0.81 ITK (0.53) BTKCLK2ITKKITSRC
SCHEMBL13894056 0.80 BTK (0.68) BTKCLK2ITKSRCFLT3
SCHEMBL105668 0.78 BTK (0.83) BTKCLK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009053269-A1 NOVEL KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2009-04-30 WO disclosed