SCHEMBL13895262

SCHEMBL13895262

C[C@@H]1[C@H](C)N(c2ccc(C(F)(F)F)cn2)CCN1S(=O)(=O)c1ccc2c(c1)C(CC(=O)O)CS2

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 5/20 0.38
NR1H3 Q13133 5/20 0.38
GPR119 Q8TDV5 1/20 0.37
GCKR Q14397 3/20 0.35
PKM P14618 1/20 0.35
CXCR3 P49682 6/20 0.35
KDM4E B2RXH2 1/20 0.35
CNR2 P34972 2/20 0.34
SGPL1 O95470 1/20 0.34
CNR1 P21554 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5778752 0.79 NR1H2 (0.40) NR1H2NR1H3GPR119GCKRCXCR3
SCHEMBL12749864 0.78 NR1H2 (0.38) NR1H2NR1H3GPR119PKMCXCR3
SCHEMBL1471200 0.78 NR1H2 (0.38) NR1H2NR1H3GPR119PKMCXCR3
SCHEMBL5746016 0.78 NR1H2 (0.46) NR1H2NR1H3GPR119SGPL1
SCHEMBL12749863 0.78 GPR119 (0.41) NR1H2NR1H3GPR119GCKRCXCR3
SCHEMBL1470499 0.78 GPR119 (0.41) NR1H2NR1H3GPR119GCKRCXCR3
SCHEMBL5768967 0.76 PPARG (0.41) NR1H2NR1H3GPR119KDM4ECNR2
SCHEMBL20308934 0.74 HMOX1 (0.38) NR1H2NR1H3GPR119GCKRCXCR3
SCHEMBL13940340 0.72 HMOX1 (0.37) NR1H2NR1H3GPR119GCKRCXCR3
SCHEMBL12828183 0.68 TBXA2R (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7517884-B2 {5-[4-(4-Trifluoromethyl-phenyl)-piperazine-1-sulfonyl]-indan-2-yl}-acetic acid; peroxisome proliferator activated receptors modulator; antidiabetic, antiinflammatory agent; obesity, hyperinsulinemia, metabolic syndrome X, polycystic ovary syndrome, ischemia-associated organ injury, diabetes KALYPSYS INC. (US) 2009-04-14 US disclosed