SCHEMBL138953

SCHEMBL138953

NCc1cccc(O)c1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29598265 1.00
Hydrochloric Acid SCHEMBL928401 0.98 ENPP2 (0.95)
Bromide SCHEMBL920224 0.98 ENPP2 (0.95)
Hydrochloric Acid SCHEMBL3564737 0.95 ENPP2 (0.91)
Hydrochloric Acid SCHEMBL18641325 0.89 ENPP2 (0.80)
Acetic Acid SCHEMBL4083695 0.88 ENPP2 (0.77)
SCHEMBL2948809 0.87 ENPP2 (0.76)
Benzylamine SCHEMBL5930798 0.82 LOXL2 (0.74)
SCHEMBL27575536 0.82 ENPP2 (0.68)
SCHEMBL29465557 0.81 TAAR1 (1.00)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 972 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118929620-A Preparation method of phenolic resin-based hard carbon nanospheres with adjustable particle size and carbon structure 北京化工大学 2024-11-12 CN claimed
CN-115228290-A Preparation method of cleaning-resistant reverse osmosis membrane 万华化学集团股份有限公司 2022-10-25 CN claimed
US-20220112156-A1 ADAMANTANECARBOXYLIC ACID BENZYL AMIDE DERIVATIVE COMPOUND AND SKIN WHITENING COMPOSITION COMPRISING SAME AMOREPACIFIC CORPORATION (KR) 2022-04-14 US claimed
CN-113286779-A Adamantane carboxylic acid benzylamide derivative compound and skin whitening composition containing same 株式会社爱茉莉太平洋 2021-08-20 CN claimed
CN-113046734-A Bivalent palladium complex solution and preparation method and application thereof 上海天承化学有限公司 2021-06-29 CN claimed
WO-2020141927-A1 ADAMANTANECARBOXYLIC ACID BENZYL AMIDE DERIVATIVE COMPOUND AND SKIN WHITENING COMPOSITION COMPRISING SAME ㈜아모레퍼시픽 2020-07-09 WO claimed
EP-3394027-B1 METHOD FOR PREPARING PHENOLICS USING A CATALYST TNO (NL) 2020-02-19 EP claimed
US-10407376-B2 Method to prepare phenolics from biomass NEDERLANDSE ORGANISATIE VOOR TOEGEPAST-NATUURWETENSCHAPPELIJK ONDERZOEK TNO (NL) 2019-09-10 US claimed
US-10364203-B2 Method for preparing phenolics using a catalyst NEDERLANDSE ORGANISATIE VOOR TOEGEPAST-NATUURWETENSCHAPPELIJK ONDERZOEK TNO (NL) 2019-07-30 US claimed
CN-109312476-A Deoxidant for boiler and deoxidization method for boiler water system 栗田工业株式会社 2019-02-05 CN claimed
WO-2000047578-A1 HETEROARYL AMIDINES, METHYLAMIDINES AND GUANIDINES AS PROTEASE INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO claimed
WO-2000044750-A1 PURINE INHIBITORS OF CYCLIN DEPENDENT KINASE 2 AND Iλ-A$g(a) CV THERAPEUTICS, INC. (US) 2000-08-03 WO claimed
EP-1021186-A4 PURINE INHIBITORS OF CYCLIN DEPENDENT KINASE 2 AND IkappaB-alpha CV THERAPEUTICS INC (US) 2000-07-26 EP claimed
EP-1021186-A1 PURINE INHIBITORS OF CYCLIN DEPENDENT KINASE 2 AND IkappaB-alpha CV THERAPEUTICS, INC. (US) 2000-07-26 EP claimed
EP-0998946-A1 Non-porphyrin compound for use as a diagnosticum and/or pharmaceutical K.U. LEUVEN RESEARCH & DEVELOPMENT (BE) 2000-05-10 EP claimed
WO-2000009169-A1 NON-PORPHYRIN COMPOUND FOR USE AS A DIAGNOSTICUM AND/OR PHARMACEUTICAL K.U. LEUVEN RESEARCH & DEVELOPMENT (BE) 2000-02-24 WO claimed
EP-0874847-A1 NOVEL PURINE DERIVATIVES HAVING, IN PARTICULAR, ANTIPROLIFERATIVE PROPERTIES, AND BIOLOGICAL USES THEREOF CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 1998-11-04 EP claimed
WO-1998005335-A9 PURINE INHIBITORS OF CYCLIN DEPENDENT KINASE 2 AND IλB-$g(a) 1998-05-28 WO claimed
WO-1998005335-A1 PURINE INHIBITORS OF CYCLIN DEPENDENT KINASE 2 AND IλB-$g(a) CV THERAPEUTICS, INC. (US) 1998-02-12 WO claimed
WO-1997020842-A1 NOVEL PURINE DERIVATIVES HAVING, IN PARTICULAR, ANTIPROLIFERATIVE PROPERTIES, AND BIOLOGICAL USES THEREOF CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (C.N.R.S.) (FR) 1997-06-12 WO claimed