SCHEMBL13902876

SCHEMBL13902876

C[C@H]([C@@H](C)O)N(C)CC#Cc1cc2c(c(C(=O)N[C@@H](CO)Cc3c[nH]c4ccccc34)c1)OCCCC2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
TACR1 P25103 2/20 0.35
ECE1 P42892 1/20 0.35
SNCA P37840 5/20 0.35
USP2 O75604 1/20 0.35
MAPK1 P28482 1/20 0.35
HTR1A P08908 1/20 0.34
SLC6A4 P31645 1/20 0.34
GHSR Q92847 1/20 0.33
MME P08473 1/20 0.33
ACE P12821 1/20 0.33
HDAC3 O15379 2/20 0.33
HDAC4 P56524 2/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC7 Q8WUI4 2/20 0.33
HDAC2 Q92769 2/20 0.33
HDAC10 Q969S8 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13962656 1.00 ALDH1A1 (0.36) ALDH1A1POLBMAPTHPGDTACR1
SCHEMBL13962172 0.92 ALDH1A1 (0.38) ALDH1A1POLBMAPTHPGDTACR1
SCHEMBL13902868 0.92 ALDH1A1 (0.38) ALDH1A1POLBMAPTHPGDTACR1
SCHEMBL13902865 0.89 ECE1 (0.38) ALDH1A1POLBMAPTHPGDTACR1
SCHEMBL13902867 0.89 ACHE (0.43) ALDH1A1POLBMAPTHPGDTACR1
SCHEMBL13902869 0.89 ALDH1A1 (0.36) ALDH1A1POLBMAPTHPGDTACR1
SCHEMBL13902864 0.88 ECE1 (0.40) ALDH1A1POLBMAPTHPGDTACR1
SCHEMBL13960314 0.87 ECE1 (0.39) ALDH1A1POLBMAPTHPGDECE1
SCHEMBL13902875 0.87 ECE1 (0.39) ALDH1A1POLBMAPTHPGDECE1
SCHEMBL13962655 0.86 ECE1 (0.37) ALDH1A1POLBMAPTHPGDTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090075987-A1 ALKYLACETYLENE SUBSTITUTED ACYLTRYPTOPHANOLS BAYER SCHERING PHARMA AG (DE) 2009-03-19 US disclosed
US-20090075987-A1 ALKYLACETYLENE SUBSTITUTED ACYLTRYPTOPHANOLS BAYER SCHERING PHARMA AG (DE) 2009-03-19 US disclosed
EP-2019102-A1 Alkylacetylene substituted Acyltryptophanols Bayer Schering Pharma AG (DE) 2009-01-28 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090075987-A1 ALKYLACETYLENE SUBSTITUTED ACYLTRYPTOPHANOLS FSHR, GNRHR, CYP19A1 ALDH1A1 2364/4885POLB 3538/4885MAPT 3935/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.