SCHEMBL13946121

SCHEMBL13946121

COc1ccc(-c2nc[nH]c(=O)c2N)c(OC)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
GAA P10253 1/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47
GFER P55789 1/20 0.47
CDC7 O00311 1/20 0.46
PDE2A O00408 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
CYP3A4 P08684 2/20 0.41
CYP1A1 P04798 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2E1 P05181 1/20 0.41
CYP2C8 P10632 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2A6 P11509 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP4B1 P13584 1/20 0.41
CYP2B6 P20813 1/20 0.41
CYP3A5 P20815 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14501800 0.82 ADORA2A (0.50) ALDH1A1HTTCDC7ADORA2AADORA1
SCHEMBL13946982 0.79 ALDH1A1 (0.50) ALDH1A1ADORA1KMT2AMEN1MAPT
SCHEMBL13946616 0.77 PKM (0.54) ALDH1A1GAAHTTADORA2AADORA1
SCHEMBL13946172 0.75 KMT2A (0.53) ALDH1A1KMT2AMAPTTHRBKDM4E
SCHEMBL10691876 0.74 PDE2A (0.55) ALDH1A1HTTCDC7PDE2ACYP3A4
SCHEMBL13946594 0.73 PDGFRB (0.47)
SCHEMBL13946598 0.73 KMT2A (0.43) ALDH1A1SRCKMT2AMAPTKDM4E
SCHEMBL13945492 0.72 ALDH1A1 (0.48) ALDH1A1GAAMAPK1KMT2AMEN1
SCHEMBL13945510 0.72 IDO1 (0.57) CYP1A1CYP1B1SRCKMT2AABL1
SCHEMBL29554628 0.71 PIM1 (0.54) ALDH1A1GAAHTTADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1603886-B1 4-SUBSTITUTED-5-CYANO-1H-PYRIMIDIN-6-(THI)ONES AS GSK-3 INHIBITORS VERTEX PHARMA (US) 2009-02-18 EP disclosed