SCHEMBL1395401

SCHEMBL1395401

Cc1[nH]c(C=C2C(=O)Nc3cccc(-c4ccncc4)c32)c(C)c1C(=O)N1CCN(C)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 13/20 0.52
FGFR1 P11362 10/20 0.52
MET P08581 4/20 0.52
PTK2B Q14289 2/20 0.52
MEN1 O00255 1/20 0.52
CCNE1 P24864 1/20 0.52
CDK2 P24941 1/20 0.52
RECQL P46063 1/20 0.52
KMT2A Q03164 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
FLT1 P17948 4/20 0.48
FLT3 P36888 4/20 0.46
AURKB Q96GD4 3/20 0.46
PDGFRB P09619 9/20 0.45
ALK Q9UM73 4/20 0.44
RET P07949 4/20 0.44
ABL1 P00519 2/20 0.44
EGFR P00533 1/20 0.41
PDGFRA P16234 1/20 0.41
PRKAA1 Q13131 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5830590 1.00 KDR (0.52) KDRFGFR1METPTK2BMEN1
SCHEMBL6323692 0.92 MET (0.56) KDRFGFR1METPTK2BMEN1
SCHEMBL6323687 0.92 MET (0.56) KDRFGFR1METPTK2BMEN1
SCHEMBL5830890 0.92 KDR (0.51) KDRFGFR1METPTK2BMEN1
SCHEMBL5830205 0.92 KDR (0.51) KDRFGFR1METPTK2BMEN1
SCHEMBL5830520 0.91 KDR (0.51) KDRFGFR1METPTK2BMEN1
SCHEMBL5830526 0.91 KDR (0.51) KDRFGFR1METPTK2BMEN1
SCHEMBL16090377 0.91 MET (0.54) KDRFGFR1METPTK2BMEN1
SCHEMBL6321868 0.90 KDR (0.52) KDRFGFR1METPTK2BMEN1
SCHEMBL6320753 0.90 KDR (0.57) KDRFGFR1METPTK2BMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160082015-A1 METHODS, COMPOSITIONS AND KITS FOR PROMOTING MOTOR NEURON SURVIVAL AND TREATING AND DIAGNOSING NEURODEGENERATIVE DISORDERS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2016-03-24 US disclosed
US-20120010178-A1 METHODS AND COMPOUNDS FOR TREATMENT OF NEURODEGENERATIVE DISORDERS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2012-01-12 US disclosed
WO-2010048273-A2 METHODS AND COMPOUNDS FOR TREATMENT OF NEURODEGENERATIVE DISORDERS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-04-29 WO disclosed
WO-2008021210-A2 METHODS AND COMPOSITIONS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS COMBINATORX, INCORPORATED (US) 2008-02-21 WO disclosed
US-20080044390-A1 Methods and compositions for the treatment of neurodegenerative disorders CHDI, INCORPORATED 2008-02-21 US disclosed
US-7053086-B2 4-heteroaryl-3-heteroarylidenyl-2-indolinones and their use as protein kinase inhibitors SUGEN, INC. (US) 2006-05-30 US disclosed
US-20040097497-A1 4-heteroaryl-3-heteroarylidenyl-2-indolinones and their use as protein kinase inhibitors SUGEN, INC. 2004-05-20 US disclosed
US-6635640-B2 4-heteroaryl-3-heteroarylidenyl-2-indolinones and their use as protein kinase inhibitors SUGEN, INC. 2003-10-21 US disclosed
US-20020187978-A1 4-Heteroaryl-3-heteroarylidenyl-2-indolinones and their use as protein kinase inhibitors SUGEN, INC. 2002-12-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160082015-A1 METHODS, COMPOSITIONS AND KITS FOR PROMOTING MOTOR NEURON SURVIVAL AND TREATING AND DIAGNOSING NEURODEGENERATIVE DISORDERS SMN1; SMN2, SOD1, NEFM KDR 4431/4885FGFR1 4574/4885MET 4540/4885
US-20020187978-A1 4-Heteroaryl-3-heteroarylidenyl-2-indolinones and their use as protein kinase inhibitors CDK2, CDK20, CDK3 KDR 1114/4885FGFR1 785/4885MET 1991/4885
US-20040097497-A1 4-heteroaryl-3-heteroarylidenyl-2-indolinones and their use as protein kinase inhibitors CDK2, CDK20, CDK3 KDR 1114/4885FGFR1 785/4885MET 1991/4885
US-20120010178-A1 METHODS AND COMPOUNDS FOR TREATMENT OF NEURODEGENERATIVE DISORDERS SMN1; SMN2, CLN6, SNCA KDR 4776/4885FGFR1 4449/4885MET 4418/4885
US-20080044390-A1 Methods and compositions for the treatment of neurodegenerative disorders HTT, SNCA, NLN KDR 4866/4885FGFR1 4760/4885MET 4576/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.