SCHEMBL13959638

SCHEMBL13959638

CC(C(=O)c1ccc(F)cc1F)c1ccc2nnc(C(C)(C)C)n2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 5/20 0.42
MAPK13 O15264 1/20 0.39
CES2 O00748 2/20 0.37
CES1 P23141 2/20 0.37
MET P08581 6/20 0.37
PRKD3 O94806 4/20 0.36
MAP4K4 O95819 4/20 0.36
CSNK1D P48730 4/20 0.36
EGFR P00533 3/20 0.36
PRKD2 Q9BZL6 3/20 0.36
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 2/20 0.36
HSD17B10 Q99714 2/20 0.36
RXFP1 Q9HBX9 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
HPGD P15428 1/20 0.36
MINK1 Q8N4C8 1/20 0.35
GSK3A P49840 2/20 0.35
KDR P35968 1/20 0.35
MAPK9 P45984 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4297287 0.88 MAPK14 (0.39) MAPK14MAPK13CES2CES1MET
SCHEMBL4299805 0.77 MAPK14 (0.39) MAPK14MAPK13CES2CES1MET
SCHEMBL4300045 0.74 MAPK14 (0.52) MAPK14CES2CES1METPRKD3
SCHEMBL8990691 0.74 MAPK14 (0.52) MAPK14CES2CES1METPRKD3
Hydrochloric Acid SCHEMBL3240832 0.73 MAPK14 (0.51) MAPK14CES2CES1METPRKD3
SCHEMBL12891157 0.71 ALDH1A1 (0.40) MAPK14KDM4EALDH1A1HPGDCYP1A2
SCHEMBL9057179 0.70 MAP4K4 (0.53) MAPK14MAPK13METPRKD3MAP4K4
SCHEMBL4211846 0.68 MAPK14 (0.68) MAPK14MAPK13
SCHEMBL7278127 0.68 CES2 (0.44) MAPK14CES2CES1KDM4EALDH1A1
SCHEMBL4304056 0.67 MAPK14 (0.42) MAPK14MAPK13METPRKD3MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009005675-A1 NOVEL TRIAZOLOPYRIDAZINES ABBOTT LABORATORIES (US) 2009-01-08 WO disclosed