SCHEMBL13982175

SCHEMBL13982175

Nc1cc(Cl)cc(Oc2c(C(F)F)ccc(CNC(=O)c3[nH]cnc3Cl)c2F)c1

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGES O14684 9/20 0.33
AKR1B1 P15121 1/20 0.33
LMNA P02545 1/20 0.33
EPHX2 P34913 1/20 0.31
SCN9A Q15858 1/20 0.30
ROCK2 O75116 1/20 0.30
ROCK1 Q13464 1/20 0.30
KLKB1 P03952 1/20 0.30
MAP4K1 Q92918 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13982482 0.90 AKR1B1 (0.33) PTGESAKR1B1LMNAEPHX2ROCK2
SCHEMBL13982082 0.90 LMNA (0.36) PTGESAKR1B1LMNAEPHX2ROCK2
SCHEMBL13982245 0.89 LMNA (0.34) PTGESAKR1B1LMNAEPHX2ROCK2
SCHEMBL3034302 0.88 CYP3A4 (0.41) PTGESLMNAEPHX2KLKB1
SCHEMBL13982246 0.86 PTGES (0.34) PTGESAKR1B1
SCHEMBL13982427 0.85 PTGES (0.35) PTGESSCN9A
SCHEMBL13982214 0.85 LMNA (0.36) PTGESAKR1B1LMNAEPHX2KLKB1
SCHEMBL13982258 0.85 PTGES (0.37) PTGESAKR1B1LMNAEPHX2KLKB1
SCHEMBL13982267 0.83 AKR1B1 (0.33) PTGESAKR1B1LMNAEPHX2ROCK2
SCHEMBL13982338 0.82 LMNA (0.36) PTGESAKR1B1LMNAEPHX2ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008154271-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-18 WO disclosed