SCHEMBL13983255

SCHEMBL13983255

Cc1nc2c(NC3CCOc4cccc(F)c43)cc(N3CCCC3=O)cc2[nH]1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 2/20 0.35
FFAR4 Q5NUL3 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.34
SYK P43405 1/20 0.33
NR3C1 P04150 1/20 0.33
DHODH Q02127 1/20 0.33
JAK2 O60674 1/20 0.32
JAK3 P52333 1/20 0.32
P2RX7 Q99572 3/20 0.32
ROCK2 O75116 1/20 0.32
OPRL1 P41146 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
LMNA P02545 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HTR6 P50406 1/20 0.31
TYK2 P29597 1/20 0.31
KMT2A Q03164 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13983278 0.98 DHODH (0.34) FFAR1FFAR4IRAK4SYKNR3C1
SCHEMBL13983283 0.95 JAK2 (0.33) DHODHJAK2JAK3ROCK2OPRL1
SCHEMBL13983256 0.89 P2RX7 (0.32) P2RX7
SCHEMBL13983252 0.89 TRPV1 (0.37) FFAR1FFAR4NR3C1JAK2JAK3
SCHEMBL13983263 0.87 PIK3CA (0.32) DHODHCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL13983254 0.86 TRPV1 (0.37) JAK2JAK3CYP3A4CYP2D6CYP2C9
SCHEMBL13983285 0.84
SCHEMBL13983267 0.84 TRPV1 (0.38) JAK2JAK3ROCK2
SCHEMBL13983529 0.83 FFAR1 (0.38) FFAR1FFAR4IRAK4SYKNR3C1
SCHEMBL13983561 0.81 FFAR1 (0.36) FFAR1FFAR4NR3C1DHODHJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008151927-A2 6-N-SUBSTITUTED BENZ IMIDAZOLE DERIVATIVES AS ACID PUMP ANTAGONISTS NYCOMED GMBH (DE) 2008-12-18 WO disclosed