SCHEMBL13985100

SCHEMBL13985100

O=C(Nc1ccccc1)c1ccc(NCC(F)(F)F)cc1

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.59
RAB9A P51151 3/20 0.59
PTPN1 P18031 3/20 0.58
MEN1 O00255 4/20 0.56
POLB P06746 4/20 0.56
KMT2A Q03164 4/20 0.56
KDM4E B2RXH2 2/20 0.56
SIRT1 Q96EB6 1/20 0.56
HDAC2 Q92769 1/20 0.56
HDAC8 Q9BY41 1/20 0.56
HDAC6 Q9UBN7 1/20 0.56
CACNA1B Q00975 1/20 0.53
APBA1 Q02410 1/20 0.53
TDP1 Q9NUW8 2/20 0.53
CTDSP1 Q9GZU7 1/20 0.53
FFAR1 O14842 1/20 0.51
HIF1A Q16665 1/20 0.50
EPAS1 Q99814 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14715847 0.81 PTPN1 (0.84) NPC1RAB9APTPN1MEN1POLB
SCHEMBL1542761 0.80 EPHX2 (0.46) MEN1POLBKMT2A
SCHEMBL26953087 0.79 PTPN1 (0.88) NPC1RAB9APTPN1MEN1POLB
SCHEMBL549076 0.79 ALDH1A1 (0.54) PTPN1TDP1
SCHEMBL1315526 0.79 PTPN1 (0.87) NPC1RAB9APTPN1MEN1POLB
SCHEMBL12678698 0.79 PLK1 (0.49) HDAC2HDAC8HDAC6
SCHEMBL10294646 0.79 PTPN1 (0.64) NPC1RAB9APTPN1MEN1POLB
SCHEMBL4247052 0.78 NPC1 (0.86) NPC1RAB9APTPN1MEN1KMT2A
SCHEMBL14715824 0.77 NPC1 (0.88) NPC1RAB9APTPN1MEN1POLB
SCHEMBL18103163 0.77 NPC1 (0.88) NPC1RAB9APTPN1MEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009002534-A1 IMIDAZOPYRIDINYL THIAZOLYL HISTONE DEACETYLASE INHIBITORS GILEAD COLORADO, INC. (US) 2008-12-31 WO disclosed