SCHEMBL13985178

SCHEMBL13985178

CC(C)(C)OC(=O)N1CC=C(c2cc(Cl)cc(-c3nnc(CC(=O)O)o3)c2)CC1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRM1 Q13255 10/20 0.45
GRM5 P41594 9/20 0.45
PDK4 Q16654 1/20 0.43
ATR Q13535 2/20 0.42
CYP11B2 P19099 1/20 0.41
NAMPT P43490 1/20 0.41
CNR1 P21554 2/20 0.39
ENPP2 Q13822 1/20 0.38
TRPV1 Q8NER1 1/20 0.38
CDK7 P50613 1/20 0.38
CDK13 Q14004 1/20 0.38
CDK12 Q9NYV4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lithium SCHEMBL4757819 0.99 GRM1 (0.44) GRM1GRM5PDK4ATRCYP11B2
SCHEMBL4757807 0.99 GRM1 (0.44) GRM1GRM5PDK4ATRCYP11B2
Lithium Ion SCHEMBL4757812 0.91 GRM1 (0.42) GRM1GRM5PDK4ATRCYP11B2
SCHEMBL4757015 0.90 SMN1; SMN2 (0.44) GRM1GRM5PDK4ATRCYP11B2
SCHEMBL28675404 0.80 PDK4 (0.55) GRM1GRM5PDK4CYP11B2NAMPT
SCHEMBL4755099 0.80 TRPV1 (0.36) ENPP2TRPV1
SCHEMBL4756914 0.78 CALCRL (0.67) NAMPT
SCHEMBL27025935 0.77 GRM1 (0.57) GRM1GRM5PDK4ATRCYP11B2
SCHEMBL13985212 0.77 SMN1; SMN2 (0.43) ENPP2TRPV1
SCHEMBL16000812 0.76 TRPV1 (0.54) GRM1GRM5PDK4ATRNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009000819-A1 5-PHENYL-1,3,4-OXADIAZOL-2-YL-ACETYL-4-PIPERIDINYL DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2008-12-31 WO disclosed