SCHEMBL28675404

SCHEMBL28675404

CC(C)(C)OC(=O)N1CC=C(c2cc(Cl)cc(Cl)c2)CC1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDK4 Q16654 1/20 0.55
NAMPT P43490 1/20 0.54
CNR1 P21554 2/20 0.50
GRM1 Q13255 10/20 0.49
GRM5 P41594 9/20 0.49
CYP11B2 P19099 1/20 0.48
CDK7 P50613 1/20 0.46
CDK13 Q14004 1/20 0.46
CDK12 Q9NYV4 1/20 0.46
HTR6 P50406 1/20 0.45
ESR2 Q92731 1/20 0.45
STS P08842 1/20 0.45
JAK1 P23458 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28671220 0.92 GRM1 (0.51) PDK4NAMPTCNR1GRM1GRM5
SCHEMBL31053182 0.92 GRM1 (0.51) PDK4NAMPTCNR1GRM1GRM5
SCHEMBL19703166 0.91 PDK4 (0.49) PDK4NAMPTCNR1GRM1GRM5
SCHEMBL652961 0.88 NAMPT (0.60) PDK4NAMPTCNR1GRM1GRM5
SCHEMBL13261659 0.88 PDK4 (0.56) PDK4NAMPTCNR1GRM1GRM5
SCHEMBL15534537 0.87 NAMPT (0.52) PDK4NAMPTCNR1GRM1GRM5
SCHEMBL19701849 0.87 NAMPT (0.52) PDK4NAMPTCNR1GRM1GRM5
SCHEMBL30191814 0.87 CYP11B2 (0.59) PDK4NAMPTCNR1GRM1GRM5
SCHEMBL4757771 0.86 PDK4 (0.45) PDK4NAMPTCNR1GRM1GRM5
SCHEMBL28672677 0.85 GRM1 (0.56) PDK4NAMPTGRM1GRM5CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113735825-B 1,2,3, 6-Tetrahydropyridine compound and preparation method and application thereof 成都康弘药业集团股份有限公司 2024-08-27 CN disclosed
CN-113735825-A 1,2,3, 6-tetrahydropyridine compound and preparation method and application thereof 成都康弘药业集团股份有限公司 2021-12-03 CN disclosed