SCHEMBL13985665

SCHEMBL13985665

Bc1cnc2[nH]c(-c3ccc(CN)cc3)nc2c1N1CCC(Cc2cccnc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.40
AURKA O14965 2/20 0.36
HRH3 Q9Y5N1 1/20 0.35
ADRB2 P07550 1/20 0.35
ADRB1 P08588 1/20 0.35
ADRB3 P13945 1/20 0.35
MTOR P42345 1/20 0.34
CYP2A6 P11509 1/20 0.34
PRMT5 O14744 1/20 0.34
VCP P55072 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
HTR1A P08908 1/20 0.33
HTR1D P28221 1/20 0.33
HTR1B P28222 1/20 0.33
CHRNA7 P36544 2/20 0.33
OGA O60502 1/20 0.33
GNRHR P30968 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14495854 0.86 AURKA (0.50) AURKAGNRHRCHRNB2CHRNA4
SCHEMBL210746 0.80 AURKA (0.41) AURKAMTORPRMT5CA12CA1
SCHEMBL13985591 0.79 AURKA (0.43) MAP4K4AURKACHRNB2CHRNA4
SCHEMBL210273 0.76 AURKA (0.61) AURKAGNRHR
SCHEMBL13985474 0.76 AURKA (0.52) AURKAGNRHR
SCHEMBL4789897 0.75 AURKA (0.42) AURKA
SCHEMBL14495689 0.74 AURKA (0.45) AURKAMTORGNRHRCHRNB2CHRNA4
SCHEMBL14495876 0.74 AURKA (0.49) AURKAGNRHR
SCHEMBL14495859 0.73 AURKA (0.56) AURKA
SCHEMBL14495795 0.71 AURKA (0.51) AURKAGNRHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001021-A1 IMIDAZOPYRIDINE DERIVATIVES USEFUL AS ENZYME INHIBITORS FOR THE TREATMENT OF CELL PROLIFERATIVE AND AUTOIMMUNE DISEASES CHROMA THERAPEUTICS LTD. (GB) 2008-12-31 WO disclosed