SCHEMBL4789897

SCHEMBL4789897

NCc1ccc(-c2nc3c(N4CCC(Oc5cccnc5)CC4)c(Br)cnc3[nH]2)cc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AURKA O14965 10/20 0.42
CHRM4 P08173 1/20 0.38
AOC3 Q16853 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KCNH2 Q12809 1/20 0.36
IKBKB O14920 1/20 0.36
CHUK O15111 1/20 0.36
LCK P06239 1/20 0.36
ROCK1 Q13464 1/20 0.36
LTA4H P09960 1/20 0.35
GBA1 P04062 1/20 0.35
JAK1 P23458 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL209520 0.91 AURKA (0.40) AURKACHRM4
SCHEMBL16152489 0.88 AURKA (0.38) AURKAGBA1
SCHEMBL4789145 0.86 CHRM4 (0.38) AURKACHRM4AOC3IKBKBCHUK
SCHEMBL210273 0.81 AURKA (0.61) AURKACYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL208759 0.80 CHEK2 (0.40) AURKA
SCHEMBL210746 0.79 AURKA (0.41) AURKA
SCHEMBL210407 0.79 AURKA (0.58) AURKACYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL209009 0.75 AURKA (0.53) AURKACYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL13985665 0.75 MAP4K4 (0.40) AURKA
SCHEMBL13985591 0.74 AURKA (0.43) AURKACYP1A2CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001021-A1 IMIDAZOPYRIDINE DERIVATIVES USEFUL AS ENZYME INHIBITORS FOR THE TREATMENT OF CELL PROLIFERATIVE AND AUTOIMMUNE DISEASES CHROMA THERAPEUTICS LTD. (GB) 2008-12-31 WO disclosed