SCHEMBL13985666

SCHEMBL13985666

CC(c1ccccc1)N1CCN(c2c(Cl)cnc3[nH]c(-c4ccc(N5CCNCC5)cc4)nc23)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 7/20 0.56
DGAT1 O75907 3/20 0.41
CETP P11597 1/20 0.39
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
ADORA2B P29275 1/20 0.38
PRMT5 O14744 2/20 0.37
KHK P50053 1/20 0.37
CDK9 P50750 2/20 0.37
CDC7 O00311 1/20 0.37
PIM1 P11309 1/20 0.37
KCNH2 Q12809 1/20 0.36
PARP1 P09874 1/20 0.35
CCNK O75909 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CCND3 P30281 1/20 0.35
CDK6 Q00534 1/20 0.35
MAPK8 P45983 1/20 0.35
MAPK9 P45984 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL210162 0.86 AURKA (0.75) AURKACNR1CNR2ADORA2B
SCHEMBL4820200 0.84 AURKA (0.49) AURKADGAT1PRMT5CDK9CCNK
SCHEMBL208728 0.81 AURKA (0.47) AURKAADORA2BKCNH2PARP1
SCHEMBL211374 0.79 AURKA (0.45) AURKADGAT1ADORA2BKCNH2
SCHEMBL210669 0.78 AURKA (0.48) AURKACNR1CNR2
SCHEMBL211945 0.76 AURKA (0.50) AURKACDK9CDC7PIM1KCNH2
SCHEMBL13985663 0.75 AURKA (0.48) AURKAKCNH2
SCHEMBL4789991 0.74 AURKA (0.47) AURKAADORA2B
SCHEMBL209704 0.74 AURKA (0.53) AURKAPARP1
SCHEMBL210044 0.73 AURKA (0.56) AURKADGAT1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001021-A1 IMIDAZOPYRIDINE DERIVATIVES USEFUL AS ENZYME INHIBITORS FOR THE TREATMENT OF CELL PROLIFERATIVE AND AUTOIMMUNE DISEASES CHROMA THERAPEUTICS LTD. (GB) 2008-12-31 WO disclosed