SCHEMBL4820200

SCHEMBL4820200

CC(c1ccccc1)N1CCN(c2c(Cl)cnc3[nH]c(-c4ccc(N5CCN(C(=O)OC(C)(C)C)CC5)cc4)nc23)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.49
CCNK O75909 1/20 0.45
CCNA2 P20248 1/20 0.45
CDK2 P24941 1/20 0.45
CCND3 P30281 1/20 0.45
CDK9 P50750 1/20 0.45
CDK6 Q00534 1/20 0.45
DGAT1 O75907 2/20 0.44
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
CKS1B P61024 2/20 0.41
SKP1 P63208 2/20 0.41
SKP2 Q13309 2/20 0.41
ALK Q9UM73 3/20 0.41
TBK1 Q9UHD2 6/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13985666 0.84 AURKA (0.56) AURKACCNKCCNA2CDK2CCND3
SCHEMBL209558 0.80 ALK (0.44) AURKACCNKCCNA2CDK2CCND3
SCHEMBL210162 0.79 AURKA (0.75) AURKA
SCHEMBL13985719 0.78 AURKA (0.58) AURKA
SCHEMBL13985589 0.78 AURKA (0.42) AURKACCNKCCNA2CDK2CCND3
SCHEMBL4754628 0.78 TBK1 (0.40) AURKACCNKCCNA2CDK2CCND3
SCHEMBL13985713 0.77 AURKA (0.47) AURKATBK1
SCHEMBL13985717 0.77 AURKA (0.44) AURKACCNKTBK1KIT
SCHEMBL25232158 0.77 KIT (0.49) CCNKCCNA2CDK2CCND3CDK9
SCHEMBL209864 0.76 TBK1 (0.44) AURKATBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001021-A1 IMIDAZOPYRIDINE DERIVATIVES USEFUL AS ENZYME INHIBITORS FOR THE TREATMENT OF CELL PROLIFERATIVE AND AUTOIMMUNE DISEASES CHROMA THERAPEUTICS LTD. (GB) 2008-12-31 WO disclosed
WO-2009001021-A1 IMIDAZOPYRIDINE DERIVATIVES USEFUL AS ENZYME INHIBITORS FOR THE TREATMENT OF CELL PROLIFERATIVE AND AUTOIMMUNE DISEASES CHROMA THERAPEUTICS LTD. (GB) 2008-12-31 WO disclosed