SCHEMBL13989372

SCHEMBL13989372

CC(=O)Nc1ccc(SCCC23C=CC(C)(O2)[C@@H]2C(=O)N(c4ccc(C#N)c(CF)c4)C(=O)[C@@H]23)cc1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
TP53 P04637 2/20 0.37
HPGD P15428 2/20 0.37
MAPK1 P28482 2/20 0.37
HTT P42858 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
HSD17B10 Q99714 2/20 0.37
MEN1 O00255 1/20 0.37
MAPT P10636 1/20 0.37
KMT2A Q03164 1/20 0.37
CACNA1B Q00975 5/20 0.37
APBA1 Q02410 5/20 0.37
RAB9A P51151 2/20 0.36
LMNA P02545 1/20 0.36
ATM Q13315 1/20 0.36
AR P10275 10/20 0.35
CRBN Q96SW2 1/20 0.33
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6433220 0.89 AR (0.48) AR
SCHEMBL3191022 0.89 AR (0.48) AR
SCHEMBL13482172 0.89 AR (0.48) AR
SCHEMBL13989355 0.84 AR (0.39) RAB9AARCRBN
SCHEMBL13889592 0.79 CACNA1B (0.52) ALDH1A1TP53HPGDMAPK1HTT
SCHEMBL13482175 0.78 CACNA1B (0.43) ALDH1A1TP53HPGDMAPK1HTT
SCHEMBL3181672 0.77 AR (0.48) AR
SCHEMBL5239091 0.77 AR (0.48) AR
SCHEMBL13482176 0.77 AR (0.48) AR
SCHEMBL13480834 0.77 AR (0.48) AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7470797-B2 Fused heterocyclic imido and amido compounds BRISTOL-MYERS SQUIBB COMPANY (US) 2008-12-30 US disclosed