SCHEMBL13992144

SCHEMBL13992144

Cc1ccsc1-c1c2c(nc3c1C(N)C(C(N)=O)S3)CCCC2=O

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
EEF2K O00418 1/20 0.39
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13991949 0.82 ALDH1A1 (0.38) CYP1A2CYP2C9KDM4E
SCHEMBL4123645 0.69 EEF2K (0.75) EEF2KCYP1A2CYP2C9KDM4E
SCHEMBL13991924 0.64 ALDH1A1 (0.36) KDM4E
SCHEMBL30174195 0.58 EEF2K (0.41) EEF2KCYP2C9KDM4E
SCHEMBL14317334 0.56 NUDT1 (0.41) KDM4E
SCHEMBL9684673 0.55 KDM4E (0.49) EEF2KCYP1A2CYP2C9KDM4E
SCHEMBL7916071 0.54 TSHR (0.44) CYP1A2CYP2C9KDM4E
SCHEMBL15598418 0.54 KDM4E (0.52) CYP1A2CYP2C9KDM4E
SCHEMBL7917747 0.54 TSHR (0.44) CYP1A2CYP2C9KDM4E
SCHEMBL13925351 0.52 TSHR (0.42) CYP1A2CYP2C9KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7465742-B2 Heterocyclic compounds having anti-HBV activity VRX HOLDCO LLC 2008-12-16 US disclosed