SCHEMBL1399376

SCHEMBL1399376

NCCc1ccccc1Sc1c[nH]c2ccc(F)c(F)c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.47
GPR84 Q9NQS5 2/20 0.47
MPO P05164 3/20 0.40
TAAR1 Q96RJ0 3/20 0.40
HTR2C P28335 2/20 0.40
HTR1D P28221 2/20 0.40
HTR1B P28222 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2A6 P11509 1/20 0.40
NFKB1 P19838 1/20 0.40
HTR7 P34969 1/20 0.40
CTSK P43235 1/20 0.40
HTR6 P50406 1/20 0.40
CYP2A13 Q16696 1/20 0.40
TRPM8 Q7Z2W7 3/20 0.40
PMP22 Q01453 1/20 0.39
SLC6A2 P23975 1/20 0.39
HTR1A P08908 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1399250 0.85 HTR2A (0.62) HTR2AGPR84MPOTAAR1HTR2C
SCHEMBL1399369 0.84 HTR2A (0.44) HTR2AMPOTAAR1HTR2CHTR1D
SCHEMBL1399373 0.83 GPR84 (0.49) HTR2AGPR84HTR6SLC6A2KMT2A
SCHEMBL4633056 0.81 HTR2A (0.45) HTR2AMPOTAAR1HTR2CHTR1D
SCHEMBL1399149 0.79 HTR2C (0.63) HTR2AMPOTAAR1HTR2CHTR1D
SCHEMBL1399316 0.79 IDO1 (0.47) HTR2AGPR84MPOTAAR1HTR2C
SCHEMBL1399370 0.79 HTR2A (0.47) HTR2AMPOTAAR1HTR2CHTR1D
SCHEMBL1399332 0.78 MPO (0.62) HTR2AGPR84MPOTAAR1HTR2C
SCHEMBL4632768 0.77 HTR2A (0.47) HTR2AGPR84MPOTAAR1HTR2C
SCHEMBL1399345 0.77 HTR2A (0.50) HTR2AMPOTAAR1HTR2CHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1860100-B1 2-(1H-indolylsulfanyl)-benzyl amine derivatives as SSRI LUNDBECK & CO AS H (DK) 2011-03-02 EP claimed