SCHEMBL1400944

SCHEMBL1400944

CCCCCCCC(C)C(=O)NCc1cc(-c2ccc(CCC(=O)O)cc2OCC(C)C)cs1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 3/20 0.38
RXRA P19793 1/20 0.37
S1PR5 Q9H228 2/20 0.36
TRPV1 Q8NER1 2/20 0.35
CYP3A4 P08684 3/20 0.34
CYP2C8 P10632 3/20 0.34
CYP2C9 P11712 3/20 0.34
CYP2B6 P20813 3/20 0.34
CYP2C19 P33261 3/20 0.34
HTR1A P08908 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2A6 P11509 2/20 0.34
CYP1A2 P05177 2/20 0.34
LTA4H P09960 2/20 0.34
CYP2E1 P05181 1/20 0.34
FFAR4 Q5NUL3 1/20 0.33
HPGD P15428 1/20 0.33
THRA P10827 1/20 0.33
THRB P10828 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL67071 0.94 RXRA (0.42) S1PR1RXRAS1PR5TRPV1CYP3A4
SCHEMBL69551 0.93 TRPV1 (0.36) TRPV1CYP3A4CYP2C8CYP2C9CYP2B6
SCHEMBL67083 0.88 PPARG (0.43) S1PR1RXRAS1PR5TRPV1HPGD
SCHEMBL70090 0.87 PPARG (0.39) TRPV1CYP3A4CYP2C8CYP2C9CYP2B6
SCHEMBL68746 0.84 MMP2 (0.40) S1PR1RXRAFFAR4HPGD
SCHEMBL1400940 0.82 S1PR1 (0.40) S1PR1RXRAS1PR5CYP3A4CYP2C8
SCHEMBL68467 0.79 RXRA (0.41) S1PR1RXRATRPV1CYP3A4CYP2C8
SCHEMBL69550 0.75 CYP3A4 (0.37) CYP3A4CYP2C8CYP2C9CYP2B6CYP2C19
SCHEMBL67800 0.75 CYP4F2 (0.39) TRPV1HPGD
SCHEMBL67070 0.75 RXRA (0.44) S1PR1RXRAS1PR5CYP3A4CYP2C8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1814871-B1 COMPOUNDS THAT MODULATE PPARY TYPE RECEPTORS, AND USE THEREOF IN COSMETIC OR PHARMACEUTICAL COMPOSITIONS GALDERMA RES & DEV (FR) 2011-03-02 EP claimed