SCHEMBL14014208

SCHEMBL14014208

COc1cccc(-c2cc(-c3ccc(Cl)cc3Cl)nc3cc(C(=O)O)nn23)c1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.52
ALDH1A1 P00352 2/20 0.52
MARS1 P56192 7/20 0.50
MAPT P10636 3/20 0.49
LMNA P02545 1/20 0.49
TP53 P04637 2/20 0.47
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
HPGD P15428 1/20 0.44
CYP2C19 P33261 1/20 0.44
NSD2 O96028 1/20 0.44
NSD1 Q96L73 1/20 0.44
NSD3 Q9BZ95 1/20 0.44
LPAR5 Q9H1C0 1/20 0.44
HPSE Q9Y251 1/20 0.44
GAA P10253 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ALDH1A3 P47895 1/20 0.41
JAK2 O60674 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14014210 0.89 MARS1 (0.63) KDM4EALDH1A1MARS1MAPTLMNA
SCHEMBL14014206 0.89 KDM4E (0.59) KDM4EALDH1A1MARS1MAPTTP53
SCHEMBL14014246 0.88 KDM4E (0.59) KDM4EALDH1A1MAPTLMNATP53
SCHEMBL14014191 0.88 KDM4E (0.62) KDM4EALDH1A1MAPTLMNATP53
SCHEMBL14014202 0.87 ALDH1A1 (0.69) KDM4EALDH1A1MARS1MAPTTP53
SCHEMBL14014295 0.86 BACE1 (0.58) KDM4EALDH1A1MARS1CYP2C9HPGD
SCHEMBL14014203 0.85 KDM4E (0.55) KDM4EALDH1A1MARS1MAPTTP53
SCHEMBL14014212 0.85 ALDH1A1 (0.66) KDM4EALDH1A1MARS1MAPTTP53
SCHEMBL14014254 0.85 KDM4E (0.73) KDM4EALDH1A1MAPTLMNATP53
SCHEMBL14014211 0.84 KDM4E (0.57) KDM4EALDH1A1MARS1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7449488-B2 Pyrazolopyrimidines as protein kinase inhibitors SCHERING CORPORATION (US) 2008-11-11 US disclosed
US-7449488-B2 Pyrazolopyrimidines as protein kinase inhibitors SCHERING CORPORATION (US) 2008-11-11 US disclosed
US-7196111-B2 Pyrazolo[1,5a]pyrimidine compounds as antiviral agents SCHERING CORPORATION (US) 2007-03-27 US disclosed
US-7196111-B2 Pyrazolo[1,5a]pyrimidine compounds as antiviral agents SCHERING CORPORATION (US) 2007-03-27 US disclosed