SCHEMBL14017263

SCHEMBL14017263

CCc1ccn2ncnc(Oc3ccc(N)cc3)c12

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.38
KDR P35968 3/20 0.36
MET P08581 5/20 0.36
TSHR P16473 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
NTRK1 P04629 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14579509 0.73 KDR (0.42) MAPTKDRTDP1
SCHEMBL14252959 0.71 MAP4K4 (0.62) TSHRTDP1
SCHEMBL18033869 0.69 EGFR (0.35) KDR
SCHEMBL4278057 0.68 KDR (0.60) KDR
SCHEMBL14017264 0.67 ERBB2 (0.38) KDRTSHR
SCHEMBL12872519 0.66 ALDH1A1 (0.44) MAPTTSHRTDP1
SCHEMBL4047329 0.64 MET (0.59) KDRMET
SCHEMBL1962838 0.63 AXL (0.38) MET
SCHEMBL12872522 0.62 ALDH1A1 (0.47) MAPTKDRTSHRTDP1
SCHEMBL15221821 0.62 FGFR1 (0.39) KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7439246-B2 Fused heterocyclic kinase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2008-10-21 US disclosed
US-7432373-B2 Processes and intermediates useful for preparing fused heterocyclic kinase inhibitors BRISTOL-MEYERS SQUIBB COMPANY (US) 2008-10-07 US disclosed
US-7348325-B2 Pyrrolotriazine kinase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2008-03-25 US disclosed
US-20070123534-A1 Pyrrolotriazine kinase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2007-05-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070123534-A1 Pyrrolotriazine kinase inhibitors MAP3K15, MAP3K5, STK25 MAPT 1469/4885KDR 1433/4885MET 1979/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.