SCHEMBL14019129

SCHEMBL14019129

CSc1nc(Cl)c2c(-c3ccccc3)n[nH]c2n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.48
DCUN1D1 Q96GG9 2/20 0.45
NPSR1 Q6W5P4 1/20 0.43
NTRK1 P04629 1/20 0.40
PPARG P37231 1/20 0.40
METAP2 P50579 1/20 0.39
NPC1 O15118 1/20 0.38
XBP1 P17861 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
PAX8 Q06710 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 1/20 0.38
PDE5A O76074 1/20 0.38
PDE1A P54750 1/20 0.38
PDE1B Q01064 1/20 0.38
PDE3B Q13370 1/20 0.38
PDE1C Q14123 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4014901 0.83 HSP90AA1 (0.45) KDM4EDCUN1D1NPSR1PPARGMETAP2
SCHEMBL5787312 0.82 HPGD (0.41) KDM4ENPSR1NTRK1NPC1RAB9A
SCHEMBL14019132 0.81 SMN1; SMN2 (0.48) KDM4EDCUN1D1NPSR1NTRK1METAP2
SCHEMBL5786736 0.80 ALDH1A1 (0.46) KDM4ENPSR1NPC1RAB9AKMT2A
SCHEMBL3393329 0.78 HPGD (0.44) KDM4ENPSR1NPC1HTTRAB9A
SCHEMBL2599336 0.74 NTRK1 (0.51) KDM4EDCUN1D1NPSR1NTRK1METAP2
SCHEMBL1950195 0.73 PPARG (0.32) PPARGRAB9ACYP1A2CYP2C9CYP2C19
SCHEMBL14441710 0.72 IDO1 (0.42) NPSR1HPGDIDO1
SCHEMBL31714660 0.72 PPARG (0.32) PPARGCYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL4844072 0.71 KDM4E (0.49) KDM4EDCUN1D1NPSR1PPARGNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7435731-B2 Substituted pyrazolo[3,4-d]pyrimadines and methods of using the same ROCHE PALO ALTO LLC (US) 2008-10-14 US disclosed