SCHEMBL14036208

SCHEMBL14036208

CC1CC(Nc2ncnc3[nH]ncc23)C1

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.68
PDPK1 O15530 2/20 0.58
ALDH1A1 P00352 1/20 0.51
PAK1 Q13153 10/20 0.49
CYP1A2 P05177 2/20 0.48
MAPK1 P28482 1/20 0.48
PTK2 Q05397 1/20 0.47
CYP2D6 P10635 1/20 0.46
KCNH2 Q12809 1/20 0.46
GRIN2B Q13224 1/20 0.46
RET P07949 1/20 0.46
PI4KA P42356 1/20 0.46
XDH P47989 1/20 0.46
LRRK2 Q5S007 1/20 0.46
PI4K2B Q8TCG2 1/20 0.46
PI4K2A Q9BTU6 1/20 0.46
PI4KB Q9UBF8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6128742 0.81 HPGDS (0.71) HPGDSPDPK1ALDH1A1PAK1CYP1A2
SCHEMBL8291809 0.81 HPGDS (1.00) HPGDSPDPK1PAK1CYP2D6KCNH2
SCHEMBL8291817 0.79 HPGDS (0.97) HPGDSPDPK1PAK1CYP2D6KCNH2
SCHEMBL14036252 0.79 HPGDS (0.60) HPGDSPDPK1ALDH1A1PAK1PTK2
SCHEMBL14621425 0.78 HPGDS (0.67) HPGDSPDPK1PAK1PTK2CYP2D6
SCHEMBL8291816 0.78 HPGDS (0.67) HPGDSPDPK1PAK1PTK2CYP2D6
SCHEMBL8291844 0.77 HPGDS (0.75) HPGDSPDPK1PAK1CYP2D6KCNH2
SCHEMBL17545974 0.76 HPGDS (0.68) HPGDSPDPK1ALDH1A1PAK1MAPK1
SCHEMBL8293284 0.76 HPGDS (0.73) HPGDSPDPK1PAK1CYP2D6KCNH2
SCHEMBL17545983 0.76 HPGDS (0.68) HPGDSPDPK1ALDH1A1PAK1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7452893-B2 4-cycloakylaminopyrazolo pyrimidine NMDA/NR2B antagonists MERCK & CO., INC. (US) 2008-11-18 US disclosed