SCHEMBL14036252

SCHEMBL14036252

C[C@H]1CC[C@H](Nc2ncnc3[nH]ncc23)CC1F

nearest known ligand 0.60

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.60
PDPK1 O15530 1/20 0.49
PAK1 Q13153 10/20 0.46
GRIN2B Q13224 6/20 0.46
KCNH2 Q12809 2/20 0.46
CYP2D6 P10635 1/20 0.46
ALDH1A1 P00352 1/20 0.44
PTK2 Q05397 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14621425 0.84 HPGDS (0.67) HPGDSPDPK1PAK1GRIN2BKCNH2
SCHEMBL8291816 0.84 HPGDS (0.67) HPGDSPDPK1PAK1GRIN2BKCNH2
SCHEMBL14036208 0.79 HPGDS (0.68) HPGDSPDPK1PAK1GRIN2BKCNH2
SCHEMBL8291809 0.76 HPGDS (1.00) HPGDSPDPK1PAK1GRIN2BKCNH2
SCHEMBL8291844 0.75 HPGDS (0.75) HPGDSPDPK1PAK1GRIN2BKCNH2
SCHEMBL8291817 0.75 HPGDS (0.97) HPGDSPDPK1PAK1GRIN2BKCNH2
SCHEMBL8293592 0.73 SLC29A1 (0.50) HPGDSPAK1GRIN2BKCNH2CYP2D6
SCHEMBL8293452 0.73 SLC29A1 (0.50) HPGDSPAK1GRIN2BKCNH2CYP2D6
SCHEMBL8293768 0.73 SLC29A1 (0.50) HPGDSPAK1GRIN2BKCNH2CYP2D6
SCHEMBL8291847 0.73 SLC29A1 (0.50) HPGDSPAK1GRIN2BKCNH2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7452893-B2 4-cycloakylaminopyrazolo pyrimidine NMDA/NR2B antagonists MERCK & CO., INC. (US) 2008-11-18 US disclosed