SCHEMBL14042267

SCHEMBL14042267

Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1NC(=O)c1ccc2nc(NC(=O)Nc3cccnc3)sc2c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 4/20 0.67
MAPK14 Q16539 3/20 0.61
KIT P10721 2/20 0.61
KDR P35968 1/20 0.61
LCK P06239 3/20 0.59
SRC P12931 2/20 0.59
BRAF P15056 6/20 0.59
DDR1 Q08345 3/20 0.58
DDR2 Q16832 3/20 0.58
POLB P06746 2/20 0.55
HTT P42858 1/20 0.55
KDM4E B2RXH2 2/20 0.53
MAPT P10636 2/20 0.53
EPHX2 P34913 1/20 0.53
EPHB2 P29323 2/20 0.53
ATM Q13315 2/20 0.53
ESYT2 A0FGR8 1/20 0.52
HACL2 A1L0T0 1/20 0.52
NBAS A2RRP1 1/20 0.52
GTPBP10 A4D1E9 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14042252 0.95 BRAF (0.66) CSF1RMAPK14KITKDRLCK
SCHEMBL4746517 0.88 LCK (0.63) CSF1RMAPK14KITKDRLCK
SCHEMBL14042248 0.88 BRAF (0.68) CSF1RMAPK14KITKDRLCK
SCHEMBL14042471 0.87 LCK (0.65) CSF1RMAPK14KITKDRLCK
SCHEMBL14042454 0.87 CSNK1D (0.66) CSF1RMAPK14KITKDRLCK
SCHEMBL14042259 0.86 BRAF (0.62) CSF1RMAPK14KITLCKSRC
SCHEMBL4863711 0.86 LCK (0.57) CSF1RMAPK14KITKDRLCK
SCHEMBL14042261 0.86 LCK (0.57) CSF1RMAPK14KITKDRLCK
SCHEMBL14042254 0.85 LCK (0.56) CSF1RMAPK14KITKDRLCK
SCHEMBL14042467 0.84 LCK (0.61) CSF1RMAPK14KITKDRLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008124393-A1 BENZOTHIAZOLE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2008-10-16 WO disclosed