SCHEMBL14044179

SCHEMBL14044179

CCCNc1nc2cc(C(F)(F)F)ccc2n2ccnc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 5/20 0.48
IKBKB O14920 1/20 0.41
HTR3E A5X5Y0 2/20 0.41
HTR3B O95264 2/20 0.41
HTR3A P46098 2/20 0.41
HTR3D Q70Z44 2/20 0.41
HTR3C Q8WXA8 2/20 0.41
HTR1D P28221 2/20 0.41
HTR2C P28335 2/20 0.41
KDM4E B2RXH2 2/20 0.41
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
HTR1A P08908 1/20 0.41
CYP2D6 P10635 1/20 0.41
TSHR P16473 1/20 0.41
NFKB1 P19838 1/20 0.41
CYP2C19 P33261 1/20 0.41
THPO P40225 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3495173 0.87 MAPK8 (0.47) MAPK8IKBKBHTR3EHTR3BHTR3A
SCHEMBL17895234 0.84 IKBKB (0.57) MAPK8IKBKBHTR3EHTR3BHTR3A
SCHEMBL8103067 0.79 MAPK8 (0.73) MAPK8IKBKBHTR3EHTR3BHTR3A
SCHEMBL3498276 0.75 KDM4E (0.42) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL17895304 0.75 IKBKB (0.68) MAPK8IKBKB
SCHEMBL31746824 0.74 ABL1 (0.43)
SCHEMBL14044186 0.74 IKBKB (0.42) IKBKBLMNAMEN1KMT2ARXFP1
SCHEMBL3496156 0.73 HTR3E (0.52) MAPK8IKBKBHTR3EHTR3BHTR3A
SCHEMBL31746683 0.72 CNR1 (0.43) MAPK8IKBKBKDM4ETP53LMNA
SCHEMBL11500648 0.71 MAPK8 (0.68) MAPK8IKBKBHTR3EHTR3BHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008117225-A2 NEW IMIDAZOLO-HETEROARYL DERIVATIVES WITH ANTIBACTERIAL PROPERTIES MUTABILIS SA (FR) 2008-10-02 WO disclosed