SCHEMBL14048355

SCHEMBL14048355

Cc1cccc(C2(N)N=N2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 4/20 0.46
HTR2C P28335 2/20 0.41
HTR2A P28223 1/20 0.41
BACE1 P56817 1/20 0.41
TP53 P04637 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
LMNA P02545 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ALDH1A1 P00352 1/20 0.38
MAPK1 P28482 1/20 0.38
HDAC4 P56524 1/20 0.38
NPC1 O15118 1/20 0.38
CASP3 P42574 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
RAB9A P51151 1/20 0.37
PARP1 P09874 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
CHRNA1 P02708 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11971724 0.74 ACHE (0.46) ACHEHTR2CHTR2AHDAC4
SCHEMBL3123866 0.74 ACHE (0.46) ACHEHTR2CHTR2ABACE1TP53
Hydrochloric Acid SCHEMBL31486432 0.72 HTR2C (0.47) ACHEHTR2CHTR2A
SCHEMBL17315641 0.71
SCHEMBL18769426 0.71
SCHEMBL13061001 0.69
Hydrochloric Acid SCHEMBL18742464 0.69
SCHEMBL4592879 0.67 ACHE (0.38) ACHEHTR2CHTR2ABACE1LMNA
M-Xylene SCHEMBL27293588 0.67 ACHE (0.86) ACHETP53TDP1LMNANPSR1
M-Xylene SCHEMBL27382740 0.67 ACHE (0.86) ACHETP53TDP1LMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1749011-B1 BICYCLIC HETEROCYCLES AS HIV INTEGRASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2008-10-29 EP disclosed