SCHEMBL4592879

SCHEMBL4592879

Cc1cccc(C2(C(Cl)(Cl)C3(c4cccc(C)c4)N=NN=N3)N=NN=N2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.38
HTR2C P28335 2/20 0.36
HTR2A P28223 1/20 0.36
LMNA P02545 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HDAC4 P56524 1/20 0.33
BACE1 P56817 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
HTT P42858 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPK1 P28482 1/20 0.32
CHRNA1 P02708 1/20 0.32
CHRNG P07510 1/20 0.32
CHRNB1 P11230 1/20 0.32
CHRNB2 P17787 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4594159 0.79 ACHE (0.35) ACHELMNAMAPTHTTALDH1A1
SCHEMBL4593434 0.78 TSHR (0.35) TAAR1
SCHEMBL2525541 0.74 ADRA2A (0.47) ACHEHTR2CHTR2ALMNANPSR1
SCHEMBL3123866 0.67 ACHE (0.46) ACHEHTR2CHTR2ALMNANPSR1
SCHEMBL14048355 0.67 ACHE (0.46) ACHEHTR2CHTR2ALMNANPSR1
SCHEMBL4593190 0.67 SLC6A3 (0.33) SLC6A2SLC6A3
SCHEMBL5280778 0.66 TSHR (0.35)
SCHEMBL11682414 0.65 CHRNA1 (0.41) ACHEHTR2CHTR2ALMNANPSR1
SCHEMBL4593654 0.64 MAOA (0.40) ALDH1A1SLC6A2SLC6A3TAAR1
SCHEMBL25839802 0.63 ACHE (0.46) ACHEHTR2CHTR2ALMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937257-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES Nederlandse Organisatie voor toegepast- natuurwetenschappelijk onderzoek TNO (NL) 2008-07-02 EP claimed
WO-2007037685-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES NEDERLANDSE ORGANISATIE VOOR TOEGEPAST-NATUURWETENSCHAPPELIJK ONDERZOEK TNO (NL) 2007-04-05 WO claimed
EP-1937257-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES Nederlandse Organisatie voor toegepast- natuurwetenschappelijk onderzoek TNO (NL) 2008-07-02 EP disclosed
WO-2007037685-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES NEDERLANDSE ORGANISATIE VOOR TOEGEPAST-NATUURWETENSCHAPPELIJK ONDERZOEK TNO (NL) 2007-04-05 WO disclosed