SCHEMBL14048846

SCHEMBL14048846

Cc1c(Cc2ccnc(N)c2)c(=O)oc2cc(O)c(I)cc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.45
GAA P10253 3/20 0.45
GLA P06280 1/20 0.45
HSD17B3 P37058 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
ERAP1 Q9NZ08 1/20 0.45
MAP2K1 Q02750 4/20 0.41
RAF1 P04049 3/20 0.41
ALDH1A1 P00352 6/20 0.41
KMT2A Q03164 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
MEN1 O00255 2/20 0.41
NQO1 P15559 3/20 0.41
POLB P06746 3/20 0.40
HPGD P15428 2/20 0.40
STS P08842 1/20 0.40
MAPT P10636 2/20 0.39
MAOB P27338 1/20 0.39
SHBG P04278 1/20 0.38
JAK2 O60674 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL961450 0.89 NQO1 (0.47) KDM4EGAAGLAHSD17B3NPSR1
SCHEMBL964530 0.87 KDM4E (0.45) KDM4EGAAGLAHSD17B3NPSR1
SCHEMBL961165 0.87 TP53 (0.49) KDM4EGAAGLAHSD17B3NPSR1
SCHEMBL959705 0.84 HSD17B3 (0.65) KDM4EGAAGLAHSD17B3NPSR1
SCHEMBL13391998 0.77 ALDH1A1 (0.54) KDM4EGAAMAP2K1RAF1ALDH1A1
SCHEMBL961790 0.75 MAP2K1 (0.60) KDM4EGAAGLAHSD17B3NPSR1
SCHEMBL960504 0.74 MAP2K1 (0.65) KDM4EGAAMAP2K1RAF1ALDH1A1
SCHEMBL959681 0.74 MAP2K1 (0.73) KDM4EGAAMAP2K1RAF1ALDH1A1
SCHEMBL959618 0.74 MAP2K1 (0.53) KDM4EGAAGLAMAP2K1RAF1
SCHEMBL963925 0.74 MAP2K1 (0.40) KDM4EGAAGLAHSD17B3NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1982982-A1 NOVEL COUMARIN DERIVATIVE HAVING ANTITUMOR ACTIVITY CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2008-10-22 EP disclosed