SCHEMBL14049583

SCHEMBL14049583

C=Cc1c2c(nn1C)N(c1ccc(C)cc1Cl)CCC2

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
BCHE P06276 1/20 0.32
TUBB4A P04350 1/20 0.31
TUBB P07437 1/20 0.31
TUBA3C P0DPH7 1/20 0.31
TUBA1B P68363 1/20 0.31
TUBA4A P68366 1/20 0.31
TUBB4B P68371 1/20 0.31
TUBB3 Q13509 1/20 0.31
TUBB2A Q13885 1/20 0.31
TUBB8 Q3ZCM7 1/20 0.31
TUBA3E Q6PEY2 1/20 0.31
TUBA1A Q71U36 1/20 0.31
TUBA1C Q9BQE3 1/20 0.31
TUBB6 Q9BUF5 1/20 0.31
TUBB2B Q9BVA1 1/20 0.31
TUBB1 Q9H4B7 1/20 0.31
PDE2A O00408 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5039786 0.91 CRHR1 (0.36) CNR1CNR2TDP1CRHR1
SCHEMBL14049584 0.82 CRHR1 (0.33) CNR1CNR2TDP1BCHETUBB4A
SCHEMBL14031301 0.82 BCHE (0.33) CNR1CNR2TDP1BCHETUBB4A
SCHEMBL5044922 0.79 CRHR1 (0.38) CNR1CNR2CRHR1
SCHEMBL5047426 0.78 CRHR1 (0.32) CRHR1
SCHEMBL5039336 0.76 CRHR1 (0.42) CNR1CNR2TDP1CRHR1
SCHEMBL5039357 0.74 CRHR1 (0.38) CNR1CNR2TDP1TUBB4ATUBB
SCHEMBL5048476 0.73 CRHR1 (0.38) CNR1CNR2CRHR1
SCHEMBL5044717 0.73 CRHR1 (0.39) CRHR1
SCHEMBL5048463 0.72 LMNA (0.38) CNR1CNR2CRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7432283-B2 Heterocyclic GABAA subtype selective receptor modulators ROCHE PALO ALTO LLC (US) 2008-10-07 US disclosed