SCHEMBL1406288

SCHEMBL1406288

O=C(O)c1c[nH]nc1C(Cl)(Cl)Cl

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.33
NOTUM Q6P988 1/20 0.33
DYRK1A Q13627 1/20 0.32
TSHR P16473 1/20 0.31
KDM5A P29375 2/20 0.31
KDM4C Q9H3R0 2/20 0.31
POLB P06746 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
KDM5B Q9UGL1 1/20 0.31
KMT2A Q03164 1/20 0.31
XDH P47989 2/20 0.30
ALOX15 P16050 1/20 0.30
F7 P08709 1/20 0.30
F3 P13726 1/20 0.30
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL783526 0.80 NOTUM (0.38) ALDH1A1NOTUMKDM5AKDM4CPOLB
SCHEMBL13373959 0.80 NOTUM (0.38) ALDH1A1NOTUMKDM5AKDM4CPOLB
Hydrochloric Acid SCHEMBL29715790 0.78 NOTUM (0.41) ALDH1A1NOTUMKDM5AKDM4CPOLB
SCHEMBL163291 0.74
SCHEMBL1406290 0.73
SCHEMBL14399039 0.72
SCHEMBL22637466 0.72 GLA (0.32) NOTUMKDM5AKDM5B
SCHEMBL2147013 0.70
SCHEMBL69630 0.70 ALDH1A1 (0.39) ALDH1A1NOTUMDYRK1ATSHRKDM5A
SCHEMBL263529 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1458670-B1 METHOD FOR PRODUCING 2-HALOGENACYL-3-AMINO-ACRYLIC ACID DERIVATIVES SALTIGO GMBH (DE) 2011-03-09 EP disclosed
EP-1458670-A1 METHOD FOR PRODUCING 2-HALOGENACYL-3-AMINO-ACRYLIC ACID DERIVATIVES Bayer Chemicals AG (DE) 2004-09-22 EP disclosed
US-6706911-B1 REACTING N-SUBSTITUTED 3-AMINOACRYLIC ESTERS WITH HALOALKYLCARBOXYLIC ANHYDRIDES IN PRESENCE OF BASE; PYRAZOLE-4-CARBOXYLIC ACID CHEMICAL INTERMEDIATES; HALOACYLATION BAYER AKTIENGESELLSCHAFT (DE) 2004-03-16 US disclosed
WO-2003051820-A1 METHOD FOR PRODUCING 2-HALOGENACYL-3-AMINO-ACRYLIC ACID DERIVATIVES BAYER CHEMICALS AG (DE) 2003-06-26 WO disclosed