SCHEMBL14065147

SCHEMBL14065147

CCC(C)(NCC(C)C)c1cnc(Nc2cccc(C(F)(F)F)c2)cc1C(C)C

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.44
CNR2 P34972 4/20 0.42
MAPT P10636 2/20 0.41
KDM4E B2RXH2 3/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
GAA P10253 1/20 0.41
AURKA O14965 4/20 0.39
EGFR P00533 1/20 0.38
PRKDC P78527 1/20 0.38
IDH2 P48735 2/20 0.37
KIF11 P52732 1/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4649728 0.78 THRB (0.47) THRBCNR2MAPTKDM4EMEN1
SCHEMBL4649749 0.75 CNR2 (0.73) THRBCNR2MAPTPOLB
SCHEMBL14381794 0.75 CNR2 (0.56) THRBCNR2MAPTKDM4EMEN1
SCHEMBL4648963 0.71 KDM4E (0.46) THRBCNR2MAPTKDM4EMEN1
SCHEMBL4648965 0.69 CNR2 (0.48) THRBCNR2MAPTKDM4EMEN1
SCHEMBL5080782 0.68 CNR2 (0.77) CNR2MAPTMEN1KMT2AALDH1A1
SCHEMBL4650376 0.67 CNR2 (0.71) CNR2
SCHEMBL5212579 0.66 CNR2 (0.77) CNR2
SCHEMBL5212362 0.66 CNR2 (0.76) CNR2
SCHEMBL2739344 0.65 LMNA (0.64) THRBMEN1KMT2AAURKAEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718613-B1 PYRIDINE DERIVATIVES AND THEIR USE AS CB2 RECEPTOR MODULATORS GLAXO GROUP LTD (GB) 2008-09-03 EP disclosed