SCHEMBL14065183

SCHEMBL14065183

C/C(=C\NC=O)c1ccc(N)cc1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.39
ALDH1A1 P00352 5/20 0.38
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36
ADRB3 P13945 1/20 0.36
CRBN Q96SW2 1/20 0.36
GAA P10253 2/20 0.36
CASP1 P29466 2/20 0.35
TSHR P16473 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MAPT P10636 4/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
KDM4E B2RXH2 2/20 0.33
CYP3A4 P08684 2/20 0.33
ESR2 Q92731 1/20 0.33
PTPN1 P18031 1/20 0.33
SIGMAR1 Q99720 1/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14064841 0.81 PDE10A (0.42) PDE10AALDH1A1ADRB2ADRB1ADRB3
SCHEMBL27352743 0.77 PDE10A (0.48) PDE10AALDH1A1ADRB2ADRB1ADRB3
SCHEMBL14064972 0.77 PDE10A (0.48) PDE10AALDH1A1ADRB2ADRB1ADRB3
SCHEMBL23865472 0.76 ERCC5 (0.43) ALDH1A1TSHRL3MBTL1CYP1A2CYP2C9
SCHEMBL3030682 0.73 ALDH1A1 (0.42) PDE10AALDH1A1ADRB2ADRB1ADRB3
SCHEMBL3030686 0.73 ALDH1A1 (0.42) PDE10AALDH1A1ADRB2ADRB1ADRB3
SCHEMBL837484 0.71 ALDH1A1 (0.50) PDE10AALDH1A1ADRB2ADRB1ADRB3
SCHEMBL7186665 0.69 ALDH1A1 (0.52) PDE10AALDH1A1ADRB2ADRB1ADRB3
Acetic Acid SCHEMBL28750958 0.68 ALDH1A1 (0.57) PDE10AALDH1A1ADRB2ADRB1ADRB3
SCHEMBL14064903 0.68 PDE10A (0.42) PDE10AALDH1A1ADRB2ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1964561-A1 Inhibitors of IMPDH enzyme Vertex Pharmaceuticals Incorporated (US) 2008-09-03 EP disclosed