SCHEMBL14065202

SCHEMBL14065202

CC1(c2ccc(S(=O)(=O)Nc3ccc(Cl)cc3C(=O)c3ccccc3)cc2)CCOCC1

nearest known ligand 0.66

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.66
HTT P42858 2/20 0.66
CCR9 P51686 15/20 0.56
TP53 P04637 1/20 0.54
MAPT P10636 1/20 0.54
KMT2A Q03164 1/20 0.54
CCR2 P41597 1/20 0.50
SLC10A6 Q3KNW5 1/20 0.48
ALDH1A1 P00352 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL343280 0.91 CCR9 (0.68) LMNAHTTCCR9TP53MAPT
SCHEMBL13805783 0.90 CCR9 (0.55) LMNAHTTCCR9TP53MAPT
SCHEMBL343361 0.90 CCR9 (0.65) LMNAHTTCCR9TP53MAPT
SCHEMBL14065196 0.90 CCR9 (0.55) LMNAHTTCCR9TP53MAPT
SCHEMBL344097 0.89 CCR9 (0.71) LMNAHTTCCR9
SCHEMBL344408 0.89 LMNA (0.52) LMNAHTTCCR9TP53MAPT
SCHEMBL10249410 0.86 CCR9 (0.69) LMNAHTTCCR9TP53MAPT
SCHEMBL344087 0.86 CCR9 (0.66) LMNAHTTCCR9
SCHEMBL342947 0.86 CCR9 (0.69) LMNAHTTCCR9TP53MAPT
SCHEMBL344537 0.86 CCR9 (0.63) LMNAHTTCCR9TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7420055-B2 Antagonists of the chemokine receptor 9 (CCR9); inhibit TECK ligand; antiinflammatory agents and immunoregulators; inflammatory bowel disease; (2-phenylsulfonamidophenyl)-pyridinyl-methanones; N-[4-chloro-2(pyridine4-carbonyl)-phenyl]4-morpholin-4-yl-benzenesulfonamide CHEMOCENTRYX, INC. (US) 2008-09-02 US disclosed