SCHEMBL1406532

SCHEMBL1406532

CCOC(=O)C(=CN(CC)CC)C(=O)C(Cl)(Cl)Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 5/20 0.42
GLO1 Q04760 1/20 0.42
CYP2C9 P11712 2/20 0.39
ALDH1A1 P00352 3/20 0.38
CYP2D6 P10635 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KMT2A Q03164 6/20 0.37
MEN1 O00255 5/20 0.37
GAA P10253 3/20 0.35
DHODH Q02127 2/20 0.35
MAPT P10636 5/20 0.34
LMNA P02545 3/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
S1PR4 O95977 1/20 0.34
S1PR1 P21453 1/20 0.34
MAPK1 P28482 1/20 0.34
TSHR P16473 1/20 0.33
CYP3A4 P08684 1/20 0.33
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1406284 0.85 CYP2C9 (0.51) NPSR1GLO1CYP2C9ALDH1A1CYP2D6
SCHEMBL1406206 0.85
SCHEMBL1406245 0.83 NPSR1 (0.42) NPSR1GLO1CYP2C9ALDH1A1CYP2D6
SCHEMBL18936311 0.83 NPSR1 (0.42) NPSR1GLO1CYP2C9ALDH1A1CYP2D6
SCHEMBL18936289 0.81 NPSR1 (0.40) NPSR1GLO1CYP2C9ALDH1A1CYP2D6
SCHEMBL18936287 0.81 NPSR1 (0.40) NPSR1GLO1CYP2C9ALDH1A1CYP2D6
SCHEMBL3512466 0.79 GLO1 (0.62) NPSR1GLO1CYP2C9ALDH1A1CYP2D6
SCHEMBL18936320 0.75 NPSR1 (0.43) NPSR1GLO1CYP2C9ALDH1A1CYP2D6
SCHEMBL18936318 0.75 NPSR1 (0.43) NPSR1GLO1CYP2C9ALDH1A1CYP2D6
SCHEMBL11201754 0.73 ALDH1A1 (0.45) NPSR1GLO1CYP2C9ALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1458670-B1 METHOD FOR PRODUCING 2-HALOGENACYL-3-AMINO-ACRYLIC ACID DERIVATIVES SALTIGO GMBH (DE) 2011-03-09 EP disclosed
EP-1458670-A1 METHOD FOR PRODUCING 2-HALOGENACYL-3-AMINO-ACRYLIC ACID DERIVATIVES Bayer Chemicals AG (DE) 2004-09-22 EP disclosed
US-6706911-B1 REACTING N-SUBSTITUTED 3-AMINOACRYLIC ESTERS WITH HALOALKYLCARBOXYLIC ANHYDRIDES IN PRESENCE OF BASE; PYRAZOLE-4-CARBOXYLIC ACID CHEMICAL INTERMEDIATES; HALOACYLATION BAYER AKTIENGESELLSCHAFT (DE) 2004-03-16 US disclosed
WO-2003051820-A1 METHOD FOR PRODUCING 2-HALOGENACYL-3-AMINO-ACRYLIC ACID DERIVATIVES BAYER CHEMICALS AG (DE) 2003-06-26 WO disclosed