SCHEMBL14067288

SCHEMBL14067288

CNc1cccc(C(F)(F)F)c1C#N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 2/20 0.45
ALDH1A1 P00352 6/20 0.44
GAA P10253 4/20 0.44
KDM4E B2RXH2 4/20 0.44
HPGD P15428 2/20 0.44
MAPT P10636 1/20 0.43
MAPK1 P28482 1/20 0.43
CACNA1B Q00975 1/20 0.43
APBA1 Q02410 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
TDP1 Q9NUW8 4/20 0.41
L3MBTL1 Q9Y468 4/20 0.39
POLB P06746 1/20 0.39
TEAD1 P28347 1/20 0.38
TEAD4 Q15561 1/20 0.38
TEAD2 Q15562 1/20 0.38
P2RX7 Q99572 2/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ADORA1 P30542 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20889924 0.84 CA2 (0.38) SLC22A12ALDH1A1GAAKDM4EHPGD
SCHEMBL1906819 0.80 AR (0.43) SLC22A12ALDH1A1GAAKDM4EHPGD
SCHEMBL2418151 0.76 SLC22A12 (0.55) SLC22A12MAPTMAPK1CACNA1BAPBA1
SCHEMBL6017719 0.76 KDM4E (0.50) ALDH1A1GAAKDM4EHPGDL3MBTL1
SCHEMBL8118463 0.76 AR (0.46) SLC22A12ALDH1A1GAAKDM4EHPGD
SCHEMBL880789 0.74 ALDH1A1 (0.59) ALDH1A1GAAKDM4EHPGDMAPT
SCHEMBL11858460 0.73 SLC22A12 (0.39) SLC22A12ALDH1A1GAAKDM4EHPGD
SCHEMBL11858450 0.73 SLC22A12 (0.39) SLC22A12ALDH1A1GAAKDM4EHPGD
SCHEMBL7868327 0.73 AR (0.46) SLC22A12AR
SCHEMBL2394925 0.73 TSHR (0.40) ALDH1A1GAAKDM4EHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1325910-B1 ALIPHATIC NITROGENOUS FIVE-MEMBERED RING COMPOUNDS MITSUBISHI TANABE PHARMA CORP (JP) 2008-09-17 EP disclosed
US-7160877-B2 Aliphatic nitrogen-containing 5-membered ring compound TANABE SEIYAKU CO., LTD. (JP) 2007-01-09 US disclosed