SCHEMBL14067959

SCHEMBL14067959

CCOC(=O)CCn1c2c(c3cccc(F)c31)CN(C(=O)OCC)CC2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 2/20 0.47
SIGMAR1 Q99720 2/20 0.47
AKR1B10 O60218 1/20 0.46
AKR1B1 P15121 1/20 0.46
PTGDR2 Q9Y5Y4 5/20 0.44
CNR2 P34972 2/20 0.42
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 3/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
HDAC10 Q969S8 1/20 0.42
HTR1A P08908 1/20 0.41
CHRM5 P08912 1/20 0.41
SLC6A2 P23975 1/20 0.41
HRH2 P25021 1/20 0.41
ADRA1D P25100 1/20 0.41
HTR1B P28222 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR1E P28566 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14067788 0.90 HDAC6 (0.46) SIGMAR1CNR2ALDH1A1HDAC1HDAC6
SCHEMBL14067789 0.87 TMEM97 (0.45) TMEM97SIGMAR1AKR1B10AKR1B1PTGDR2
SCHEMBL14067833 0.83 HDAC1 (0.49) AKR1B10AKR1B1PTGDR2KDM4EHDAC1
SCHEMBL14067942 0.81 HRH1 (0.46) CNR2HDAC1HDAC6CHRM5HRH1
SCHEMBL14067970 0.81 HDAC1 (0.40) CNR2KDM4EALDH1A1HDAC1HDAC6
SCHEMBL14067777 0.81 HDAC6 (0.47) PTGDR2KDM4EALDH1A1HDAC1HDAC6
SCHEMBL14067957 0.78 HDAC1 (0.60) TMEM97SIGMAR1AKR1B10AKR1B1PTGDR2
SCHEMBL14067791 0.77 HDAC1 (0.44) CNR2ALDH1A1HDAC1HDAC6HDAC10
SCHEMBL14067786 0.76 AKR1B10 (0.55) AKR1B10AKR1B1PTGDR2CNR2HRH1
SCHEMBL23148492 0.75 PTGDR2 (0.59) AKR1B10AKR1B1PTGDR2HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008115098-A2 SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-PYRIDO[4,3-B]INDOLES, METHODS FOR THE PRODUCTION AND THE USE THEREOF ALLA CHEM, LLC (US) 2008-09-25 WO disclosed