SCHEMBL14067968

SCHEMBL14067968

CC(C)NC(=O)c1cc(F)ccc1CN

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.44
ALDH1A1 P00352 2/20 0.43
ANO1 Q5XXA6 1/20 0.40
MLYCD O95822 1/20 0.40
EIF2S1 P05198 2/20 0.39
EIF2AK3 Q9NZJ5 2/20 0.39
PSMB11 A5LHX3 1/20 0.38
PSMA7 O14818 1/20 0.38
PSMB1 P20618 1/20 0.38
PSMA1 P25786 1/20 0.38
PSMA2 P25787 1/20 0.38
PSMA3 P25788 1/20 0.38
PSMA4 P25789 1/20 0.38
PSMB8 P28062 1/20 0.38
PSMB9 P28065 1/20 0.38
PSMA5 P28066 1/20 0.38
PSMB4 P28070 1/20 0.38
PSMB6 P28072 1/20 0.38
PSMB5 P28074 1/20 0.38
PSMB10 P40306 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4762160 0.98 ALOX5 (0.43) ALOX5ALDH1A1ANO1MLYCDEIF2S1
SCHEMBL1503262 0.83 GAA (0.43) ALDH1A1GAAHPGDKEAP1
Hydrochloric Acid SCHEMBL3840135 0.81 GAA (0.42) ALDH1A1GAAHPGDKEAP1
Hydrochloric Acid SCHEMBL4763208 0.81 GAA (0.42) ALDH1A1GAAHPGDKEAP1
SCHEMBL14067872 0.80 HDAC4 (0.41) PSMB11PSMA7PSMB1PSMA1PSMA2
SCHEMBL2076694 0.80 SLC6A4 (0.44) ALDH1A1GAAHPGDKEAP1
SCHEMBL7137660 0.79 CES2 (0.55) ALOX5ALDH1A1ANO1PSMB11PSMA7
Hydrochloric Acid SCHEMBL4767213 0.79 HDAC4 (0.40) EIF2S1EIF2AK3PSMB11PSMA7PSMB1
SCHEMBL6755715 0.79 MAPK8 (0.44) KEAP1
Hydrochloric Acid SCHEMBL1977404 0.78 SLC6A4 (0.43) ALDH1A1GAAHPGDKEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1496836-B1 N-(SUBSTITUTED BENZYL)-8-HYDROXY-1,6-NAPHTHYRIDINE-7- CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2008-09-24 EP disclosed
US-7323460-B2 N-(substituted benzyl)-8-hydroxy-1,6-naphthyridine-7-carboxamides useful as HIV integrase inhibitors MERCK & CO., INC. (US) 2008-01-29 US disclosed
US-7323460-B2 N-(substituted benzyl)-8-hydroxy-1,6-naphthyridine-7-carboxamides useful as HIV integrase inhibitors MERCK & CO., INC. (US) 2008-01-29 US disclosed